SCHEMBL7254116

SCHEMBL7254116

N#CCCCBr.N#CCCCN1CCC(CNC(=O)c2cc(Cl)c(N)[nH]c2=O)CC1

nearest known ligand 0.47

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 8/20 0.44
KCNH2 Q12809 2/20 0.40
CACNA1I Q9P0X4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6329300 0.96 HTR4 (0.47) HTR4KCNH2CACNA1I
SCHEMBL7259053 0.86 HTR4 (0.46) HTR4KCNH2CACNA1I
SCHEMBL7258023 0.85 HTR4 (0.47) HTR4
SCHEMBL7259539 0.85 HTR4 (0.51) HTR4
SCHEMBL7254333 0.85 HTR4 (0.47) HTR4
SCHEMBL7260241 0.84 HTR4 (0.44) HTR4KCNH2CACNA1I
SCHEMBL7257589 0.84 HTR4 (0.49) HTR4
N-Propyl Bromide SCHEMBL7255030 0.84 HTR4 (0.46) HTR4KCNH2CACNA1I
SCHEMBL14258189 0.84 NR4A2 (0.53) HTR4
SCHEMBL6328116 0.83 HTR4 (0.49) HTR4KCNH2CACNA1I

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003057688-A2 OXO OR OXY-PYRIDINE COMPOUNDS AS 5-HT4 RECEPTOR MODULATORS PFIZER JAPAN INC. (JP) 2003-07-17 WO disclosed