SCHEMBL7254118

SCHEMBL7254118

O=c1c2c(n(-c3ccc4occc4c3)c3ccccc13)CN(c1ncc(-c3ncccn3)cn1)C2

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.34
DRD2 P14416 1/20 0.34
DRD3 P35462 1/20 0.34
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
DYRK1A Q13627 1/20 0.32
CHRNA7 P36544 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6407211 0.92 PDE5A (0.34) KCNH2DRD2DRD3DYRK1ACHRNA7
SCHEMBL7254113 0.67 PDE5A (0.59)
SCHEMBL7254126 0.64 PDE5A (0.43)
SCHEMBL15965710 0.63 GPR84 (0.40) KCNH2DRD2DRD3MAOAMAOB
SCHEMBL16452338 0.62 MKNK1 (0.34) KCNH2DRD2DRD3MAOAMAOB
SCHEMBL15964334 0.61 L3MBTL1 (0.46) DYRK1A
SCHEMBL20426812 0.60 CHRNA7 (0.35) KCNH2MAOADYRK1ACHRNA7
SCHEMBL20426625 0.60 PTPN1 (0.38) KCNH2MAOADYRK1ACHRNA7
SCHEMBL20426784 0.59 KDM4E (0.37) MAOAMAOB
SCHEMBL19849125 0.59 CHEK2 (0.34) MAOAMAOBDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6635638-B2 Treatment of sexual dysfunction, cardiovascular system disorders ORTHO-MCNEIL PHARMACEUTICAL, INC. 2003-10-21 US disclosed