SCHEMBL7254124

SCHEMBL7254124

O=C1NC2(CCCCC2=O)c2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
POLB P06746 1/20 0.43
TNKS O95271 1/20 0.42
TNKS2 Q9H2K2 1/20 0.42
AKR1B1 P15121 1/20 0.41
GRIN1 Q05586 3/20 0.40
GRIN2A Q12879 3/20 0.40
SLC6A4 P31645 2/20 0.40
GRIN2D O15399 2/20 0.40
GRIN3B O60391 2/20 0.40
GRIN2B Q13224 2/20 0.40
GRIN2C Q14957 2/20 0.40
GRIN3A Q8TCU5 2/20 0.40
OPRK1 P41145 1/20 0.40
LMNA P02545 1/20 0.40
OPRM1 P35372 1/20 0.40
CACNA1C Q13936 1/20 0.40
PDE7A Q13946 1/20 0.37
KDM4E B2RXH2 3/20 0.37
TSHR P16473 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9038579 0.84 AKR1B1 (0.56) ALDH1A1POLBAKR1B1TSHRTDP1
SCHEMBL9040587 0.79 AKR1B1 (0.61) ALDH1A1POLBAKR1B1LMNATSHR
SCHEMBL9037891 0.75 TSHR (0.59) ALDH1A1POLBAKR1B1TSHRTDP1
SCHEMBL9038575 0.75 MEN1 (0.42) ALDH1A1POLBTNKSTNKS2AKR1B1
SCHEMBL11637692 0.74 PDE7A (0.54) ALDH1A1POLBTNKSTNKS2LMNA
SCHEMBL30930016 0.73 PDE7A (0.57) ALDH1A1POLBTNKSTNKS2LMNA
SCHEMBL11641417 0.73 PDE7A (0.57) ALDH1A1POLBTNKSTNKS2LMNA
SCHEMBL30671022 0.72 ALDH1A1 (0.41) ALDH1A1POLBAKR1B1GRIN1GRIN2A
SCHEMBL28498656 0.70 GRIN1 (0.45) ALDH1A1GRIN1GRIN2ASLC6A4GRIN2D
SCHEMBL8728316 0.70 ALDH1A1 (0.45) ALDH1A1POLBAKR1B1KDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6664258-B1 Transphenylpiperazines; central dopaminergic activity PFIZER INC 2003-12-16 US disclosed