SCHEMBL9040587

SCHEMBL9040587

O=C1NC2(CCCc3ccccc32)c2ccccc21

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 7/20 0.61
CASP6 P55212 1/20 0.50
TSHR P16473 2/20 0.49
TDP1 Q9NUW8 1/20 0.49
ALDH1A1 P00352 3/20 0.45
POLB P06746 1/20 0.45
USP2 O75604 1/20 0.43
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9038579 0.95 AKR1B1 (0.56) AKR1B1CASP6TSHRTDP1ALDH1A1
SCHEMBL9037891 0.90 TSHR (0.59) AKR1B1CASP6TSHRTDP1ALDH1A1
SCHEMBL9037851 0.82 AKR1B1 (0.56) AKR1B1CASP6LMNA
SCHEMBL9038575 0.80 MEN1 (0.42) AKR1B1TDP1ALDH1A1POLBLMNA
SCHEMBL7254124 0.79 ALDH1A1 (0.43) AKR1B1TSHRTDP1ALDH1A1POLB
SCHEMBL9039157 0.78 AKR1B1 (0.53) AKR1B1POLBLMNA
SCHEMBL1395366 0.76 AKR1B1 (1.00) AKR1B1CASP6TSHRTDP1
SCHEMBL9041593 0.75 PARP1 (0.44) AKR1B1TSHRTDP1ALDH1A1POLB
SCHEMBL11379499 0.74 AKR1B1 (0.73) AKR1B1CASP6TSHRTDP1ALDH1A1
SCHEMBL11154103 0.74 AKR1B1 (0.73) AKR1B1CASP6TSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0441598-B1 Spiroisoindole compounds ZENECA INC (US) 1996-09-04 EP disclosed
US-5098925-A Neurological disorders in mammals ICI AMERICAS INC. (US) 1992-03-24 US disclosed
EP-0441598-A2 Spiroisoindole compounds ZENECA INC. (US) 1991-08-14 EP disclosed