SCHEMBL9038575

SCHEMBL9038575

O=C1NC2(CCCc3sccc32)c2ccccc21

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
ALDH1A1 P00352 3/20 0.40
LMNA P02545 2/20 0.40
HTT P42858 2/20 0.40
MAPT P10636 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
AKR1B1 P15121 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.36
POLB P06746 1/20 0.35
TNKS O95271 1/20 0.34
TNKS2 Q9H2K2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9040587 0.80 AKR1B1 (0.61) ALDH1A1LMNATDP1AKR1B1POLB
SCHEMBL9038579 0.75 AKR1B1 (0.56) ALDH1A1TDP1AKR1B1POLB
SCHEMBL7254124 0.75 ALDH1A1 (0.43) ALDH1A1LMNATDP1AKR1B1POLB
SCHEMBL9234892 0.74 AKR1B1 (0.57) MEN1KMT2ATDP1AKR1B1
SCHEMBL9037891 0.73 TSHR (0.59) ALDH1A1TDP1AKR1B1POLB
SCHEMBL9042847 0.71 AKR1B1 (0.41) MEN1KMT2AAKR1B1
SCHEMBL15606172 0.71 AKR1B1 (0.41) MEN1KMT2AALDH1A1LMNAHTT
SCHEMBL9039898 0.70 AVPR1A (0.39) MEN1KMT2AALDH1A1LMNAMAPT
SCHEMBL9041593 0.68 PARP1 (0.44) MEN1KMT2AALDH1A1MAPTTDP1
SCHEMBL30671022 0.67 ALDH1A1 (0.41) ALDH1A1TDP1AKR1B1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0441598-B1 Spiroisoindole compounds ZENECA INC (US) 1996-09-04 EP disclosed
US-5098925-A Neurological disorders in mammals ICI AMERICAS INC. (US) 1992-03-24 US disclosed
EP-0441598-A2 Spiroisoindole compounds ZENECA INC. (US) 1991-08-14 EP disclosed