SCHEMBL7256231

SCHEMBL7256231

Cc1ccc(C(=O)NC(Cc2ccccc2)c2ccccc2)c(Cl)n1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 1/20 0.53
ALDH1A1 P00352 2/20 0.51
HTT P42858 1/20 0.51
NCOA1 Q15788 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
NCOA3 Q9Y6Q9 1/20 0.51
EGFR P00533 3/20 0.51
HSD17B2 P37059 1/20 0.48
CCR3 P51677 1/20 0.43
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
HSD17B10 Q99714 1/20 0.43
GRM5 P41594 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7256356 0.82 EGFR (0.58) TACR3ALDH1A1HTTSMN1; SMN2EGFR
SCHEMBL9569932 0.81 ADORA2A (0.58) TACR3ALDH1A1EGFRKDM4ELMNA
SCHEMBL21676260 0.74 EGFR (0.54) ALDH1A1EGFRHPGDTSHR
SCHEMBL4173835 0.74 CTSV (0.53) TACR3ALDH1A1HTTNCOA1SMN1; SMN2
SCHEMBL7257209 0.74 TACR3 (0.51) TACR3ALDH1A1HTTNCOA1SMN1; SMN2
SCHEMBL19452099 0.73 TACR3 (0.50) TACR3ALDH1A1HTTNCOA1SMN1; SMN2
SCHEMBL10988800 0.72 MAPK1 (0.54) TACR3ALDH1A1HTTNCOA1SMN1; SMN2
SCHEMBL5438509 0.72 MEN1 (0.51) ALDH1A1HTTSMN1; SMN2EGFRKDM4E
SCHEMBL701920 0.71 TAS1R3 (0.48) EGFR
SCHEMBL14284682 0.71 TACR3 (0.53) TACR3ALDH1A1HTTNCOA1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030195212-A1 Novel melanocortin receptor agonists and antagonists MELACURE THERAPEUTICS AB (SE) 2003-10-16 US claimed
EP-1254114-A2 MELANOCORTIN RECEPTOR AGONISTS AND ANTAGONISTS Melacure Therapeutics AB (SE) 2002-11-06 EP claimed
WO-2001055106-A2 NOVEL MELANOCORTIN RECEPTOR AGONISTS AND ANTAGONISTS MELACURE THERAPEUTICS AB (SE) 2001-08-02 WO claimed
EP-1254114-A2 MELANOCORTIN RECEPTOR AGONISTS AND ANTAGONISTS Melacure Therapeutics AB (SE) 2002-11-06 EP disclosed
WO-2001055106-A2 NOVEL MELANOCORTIN RECEPTOR AGONISTS AND ANTAGONISTS MELACURE THERAPEUTICS AB (SE) 2001-08-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030195212-A1 Novel melanocortin receptor agonists and antagonists MC1R, MC5R, MC4R TACR3 255/4885ALDH1A1 2823/4885HTT 884/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.