SCHEMBL7256356

SCHEMBL7256356

Cc1ccc(C(=O)NC(c2ccccc2)c2ccccc2)c(Cl)n1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.58
LMNA P02545 3/20 0.47
ALDH1A1 P00352 3/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
TACR3 P29371 1/20 0.47
HSD17B2 P37059 3/20 0.44
ADORA2A P29274 1/20 0.44
ADORA1 P30542 1/20 0.44
HPGDS O60760 2/20 0.44
RXFP1 Q9HBX9 1/20 0.44
HTT P42858 2/20 0.43
MEN1 O00255 1/20 0.43
MAPT P10636 1/20 0.43
KMT2A Q03164 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9569932 0.87 ADORA2A (0.58) EGFRLMNAALDH1A1TACR3ADORA2A
SCHEMBL7256231 0.82 TACR3 (0.53) EGFRLMNAALDH1A1SMN1; SMN2TACR3
SCHEMBL21676260 0.80 EGFR (0.54) EGFRALDH1A1ADORA2AADORA1MAPT
SCHEMBL17670900 0.77 TACR3 (0.47) LMNAALDH1A1TACR3HSD17B2ADORA2A
SCHEMBL2472432 0.77 EGFR (0.50) EGFRLMNAALDH1A1ADORA2AADORA1
SCHEMBL3387703 0.77 EGFR (0.50) EGFRLMNAALDH1A1ADORA2AADORA1
SCHEMBL5438509 0.75 MEN1 (0.51) EGFRALDH1A1SMN1; SMN2RXFP1HTT
SCHEMBL6988044 0.75 EGFR (0.58) EGFRLMNAALDH1A1SMN1; SMN2MAPT
SCHEMBL14469060 0.75 EGFR (0.57) EGFRLMNAALDH1A1SMN1; SMN2
SCHEMBL701920 0.74 TAS1R3 (0.48) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030195212-A1 Novel melanocortin receptor agonists and antagonists MELACURE THERAPEUTICS AB (SE) 2003-10-16 US claimed
EP-1254114-A2 MELANOCORTIN RECEPTOR AGONISTS AND ANTAGONISTS Melacure Therapeutics AB (SE) 2002-11-06 EP claimed
WO-2001055106-A2 NOVEL MELANOCORTIN RECEPTOR AGONISTS AND ANTAGONISTS MELACURE THERAPEUTICS AB (SE) 2001-08-02 WO claimed
EP-1254114-A2 MELANOCORTIN RECEPTOR AGONISTS AND ANTAGONISTS Melacure Therapeutics AB (SE) 2002-11-06 EP disclosed
WO-2001055106-A2 NOVEL MELANOCORTIN RECEPTOR AGONISTS AND ANTAGONISTS MELACURE THERAPEUTICS AB (SE) 2001-08-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030195212-A1 Novel melanocortin receptor agonists and antagonists MC1R, MC5R, MC4R EGFR 909/4885LMNA 4570/4885ALDH1A1 2823/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.