SCHEMBL7256408

SCHEMBL7256408

COc1cccc(C(=O)c2ccc3[nH]c(=O)sc3c2)c1

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.62
PDE3A Q14432 1/20 0.62
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
STS P08842 3/20 0.49
CES2 O00748 1/20 0.49
CES1 P23141 1/20 0.49
PARP1 P09874 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
MTNR1B P49286 1/20 0.45
CYP2C8 P10632 1/20 0.44
ESR1 P03372 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
TSHR P16473 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9483327 0.88 PDE3B (0.68) PDE3BPDE3AMEN1KMT2ANPC1
SCHEMBL7257829 0.82 ESR1 (0.46) PDE3BPDE3AMEN1KMT2APARP1
SCHEMBL5727283 0.82 ESR1 (0.52) PDE3BPDE3AMEN1KMT2ANPC1
SCHEMBL5727262 0.80 POLB (0.49) PDE3BPDE3AMEN1KMT2ANPC1
SCHEMBL5726426 0.80 PGR (0.61) PDE3BPDE3AMEN1KMT2ANPC1
SCHEMBL9484835 0.79 SMN1; SMN2 (0.67) PDE3BPDE3ASMN1; SMN2CYP1A2CYP3A4
SCHEMBL1848088 0.78 PDE3B (1.00) PDE3BPDE3AMEN1KMT2ANPC1
SCHEMBL4823687 0.78 CES2 (0.77) MEN1KMT2ANPC1RAB9ASTS
SCHEMBL31414638 0.78 CES2 (0.77) MEN1KMT2ANPC1RAB9ASTS
SCHEMBL9484422 0.77 ALDH1A1 (0.50) PDE3BPDE3AMEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003027108-A1 HETEROCYCLIC DERIVATIVES AND THEIR USE AS HYPOGLYCAEMIC AND HYPOLIPIDEMIC AGENTS LES LABORATOIRES SERVIER (FR) 2003-04-03 WO disclosed