SCHEMBL7258984

SCHEMBL7258984

COc1ccc(-c2cccc(OCC[C@H](c3nc(C(N)=O)c[nH]3)[C@H](C)O)c2)cn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 2/20 0.41
CHEK1 O14757 1/20 0.41
MKNK1 Q9BUB5 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40
HSD17B1 P14061 1/20 0.39
HSD17B2 P37059 1/20 0.39
SCN9A Q15858 1/20 0.39
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
TYK2 P29597 1/20 0.39
JAK3 P52333 1/20 0.39
ADA P00813 1/20 0.38
CTSA P10619 1/20 0.37
PLCG1 P19174 1/20 0.37
FAAH O00519 4/20 0.37
LTB4R Q15722 1/20 0.35
LOXL2 Q9Y4K0 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
LRRK2 Q5S007 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7258788 0.89 CHEK2 (0.39) CHEK2CHEK1MKNK2SCN9AADA
SCHEMBL7258881 0.81 ADA (0.39) CHEK2MKNK2SCN9AJAK2ADA
SCHEMBL7258747 0.81 ADA (0.39) CHEK2CHEK1MKNK2HSD17B1HSD17B2
SCHEMBL7263018 0.79 ADA (0.41) CHEK2MKNK2HSD17B1HSD17B2JAK2
SCHEMBL7259458 0.78 ADA (0.40) CHEK2CHEK1MKNK2SCN9AADA
SCHEMBL5671212 0.78 ADA (0.63) CHEK2CHEK1MKNK1MKNK2HSD17B1
SCHEMBL7259601 0.77 ADA (0.44) ADA
SCHEMBL7264341 0.77 CHEK2 (0.35) CHEK2CHEK1MKNK2SCN9AADA
SCHEMBL7264346 0.76 ATP4A (0.38) ADA
SCHEMBL7258942 0.76 ADA (0.43) CHEK2ADA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003006437-A1 IMIDAZOLE DERIVATIVES AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-01-23 WO claimed
WO-2003006437-A1 IMIDAZOLE DERIVATIVES AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-01-23 WO disclosed