SCHEMBL7259689

SCHEMBL7259689

O=C1CCn2c(-c3ccsc3)nc3cccc1c32

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 14/20 0.47
KCNH2 Q12809 4/20 0.40
GRM2 Q14416 4/20 0.40
HTR3A P46098 1/20 0.40
PIK3CD O00329 1/20 0.37
PIK3CA P42336 1/20 0.37
PIK3CB P42338 1/20 0.37
PRKDC P78527 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6199833 0.83 PARP1 (0.66) PARP1KCNH2GRM2HTR3A
SCHEMBL8824023 0.80 PARP1 (0.68) PARP1KCNH2GRM2HTR3A
SCHEMBL423080 0.75 PARP1 (0.56) PARP1KCNH2GRM2HTR3A
SCHEMBL6139222 0.73 PARP1 (0.44) PARP1KCNH2GRM2HTR3A
SCHEMBL7265263 0.72 PARP1 (0.41) PARP1KCNH2GRM2HTR3A
Ethylene SCHEMBL6511634 0.70 PARP1 (0.42) PARP1KCNH2GRM2HTR3A
SCHEMBL7260381 0.70 NPC1 (0.46) PARP1HTR3A
SCHEMBL7265103 0.70 NPC1 (0.46) PARP1HTR3A
SCHEMBL9675375 0.69 PARP1 (0.45) PARP1KCNH2GRM2HTR3A
SCHEMBL7266288 0.69 NPC1 (0.47) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003051879-A1 KNOWN AND NOVEL 4,5-DIHYDRO-IMIDAZO[4,5,1-IJ]QUINOLIN-6-ONES USEFUL AS POLY(ADP-RIBOSE)POLYMERASE INHIBITORS ALTANA PHARMA AG (DE) 2003-06-26 WO disclosed