SCHEMBL7259758

SCHEMBL7259758

CCOC(=O)Cn1c(Cl)cnc(NC(CNCCOCCOc2ccc(Cl)cc2CNC(=O)OC(C)(C)C)CC2CC2)c1=O

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
F2 P00734 15/20 0.36
PRSS1 P07477 2/20 0.35
PRSS2 P07478 2/20 0.35
PRSS3 P35030 2/20 0.35
MASP2 O00187 1/20 0.33
ADRB2 P07550 1/20 0.32
HTR1A P08908 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
PTGER1 P34995 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7254370 0.84 F2 (0.43) F2PRSS1PRSS2PRSS3MASP2
SCHEMBL7254368 0.84 F2 (0.43) F2PRSS1PRSS2PRSS3MASP2
SCHEMBL7255198 0.76 F2 (0.46) F2PRSS1PRSS2PRSS3MASP2
SCHEMBL7255193 0.70 F2 (0.39) F2PRSS1PRSS2PRSS3MASP2
SCHEMBL30933792 0.68 CYP1A2 (0.55) ADRB2HTR1ACYP1A2CYP2D6KDM4E
SCHEMBL7254246 0.67 MEN1 (0.41) F2CYP1A2KDM4EALDH1A1MEN1
SCHEMBL7254244 0.67 MEN1 (0.41) F2CYP1A2KDM4EALDH1A1MEN1
SCHEMBL7254326 0.67 KDM4E (0.48) CYP1A2CYP2D6KDM4EALDH1A1MEN1
SCHEMBL7255220 0.67 KDM4E (0.48) KDM4EALDH1A1MEN1KMT2APTGER1
SCHEMBL7260017 0.65 KDM4E (0.46) ADRB2HTR1AKDM4EALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003011222-A2 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2003-02-13 WO disclosed