SCHEMBL7260731

SCHEMBL7260731

COC(=O)c1ccc(-c2ccc(N(Cc3cccnc3)C(=O)c3ccccc3)cc2)o1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.55
TSHR P16473 1/20 0.55
PDK1 Q15118 12/20 0.47
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 2/20 0.46
NPC1 O15118 1/20 0.46
USP2 O75604 1/20 0.46
MAPT P10636 1/20 0.46
MAPK1 P28482 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HSD17B10 Q99714 1/20 0.46
LMNA P02545 1/20 0.45
HTT P42858 1/20 0.45
CYP3A4 P08684 1/20 0.44
PTGES O14684 1/20 0.44
ALOX5 P09917 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7255144 0.90 GAA (0.59) GAATSHRPDK1ALDH1A1KDM4E
SCHEMBL7259737 0.75 FNTA (0.51)
SCHEMBL7260743 0.75 ALDH1A1 (0.57) ALDH1A1KDM4ENPC1USP2MAPT
SCHEMBL17212160 0.73 ALDH1A1 (0.53) ALDH1A1KDM4ENPC1USP2MAPT
SCHEMBL13571398 0.72 TSHR (0.84) GAATSHRPDK1NPC1RAB9A
SCHEMBL18464035 0.71 KMT2A (0.57) GAATSHRALDH1A1NPC1RAB9A
SCHEMBL18464136 0.71 TSHR (0.54) GAATSHRALDH1A1KDM4ENPC1
SCHEMBL3059132 0.70 ALDH1A1 (0.62) GAAALDH1A1KDM4ERAB9ALMNA
SCHEMBL6735689 0.69 GRM2 (0.60) GAATSHRPDK1ALDH1A1KDM4E
SCHEMBL22289326 0.69 GAA (0.73) GAATSHRALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003099812-A1 PHENYL-FURAN OR PHENYL-THIOPHENE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICINE PIERRE FABRE MEDICAMENT (FR) 2003-12-04 WO disclosed