SCHEMBL7260743

SCHEMBL7260743

COC(=O)c1ccc(-c2ccc(NCc3cccnc3)cc2)o1

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.57
KDM4E B2RXH2 2/20 0.57
LMNA P02545 1/20 0.57
CYP3A4 P08684 11/20 0.55
CYP2C9 P11712 11/20 0.55
CYP2C19 P33261 11/20 0.55
CYP1A2 P05177 7/20 0.52
CYP2D6 P10635 7/20 0.52
NPC1 O15118 2/20 0.52
MAPK1 P28482 2/20 0.52
RAB9A P51151 2/20 0.52
USP2 O75604 1/20 0.52
MAPT P10636 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
HSD17B10 Q99714 1/20 0.52
LTA4H P09960 1/20 0.50
POLB P06746 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6727719 0.81 CA1 (0.69) ALDH1A1LTA4HPOLB
SCHEMBL17212160 0.80 ALDH1A1 (0.53) ALDH1A1KDM4ELMNACYP3A4CYP2C9
SCHEMBL13766317 0.75 ALDH1A1 (0.73) ALDH1A1KDM4ECYP3A4CYP2C9CYP2C19
SCHEMBL7260731 0.75 GAA (0.55) ALDH1A1KDM4ELMNACYP3A4NPC1
SCHEMBL5440630 0.74 ALDH1A1 (0.66) ALDH1A1KDM4ELMNACYP1A2CYP2D6
SCHEMBL5735703 0.74 ABL1 (0.52) ALDH1A1KDM4ECYP2C19CYP1A2NPC1
SCHEMBL6727493 0.73 TSHR (0.58) ALDH1A1KDM4ERAB9AMAPTSMN1; SMN2
SCHEMBL2636199 0.73 LTA4H (0.67) ALDH1A1LMNACYP3A4CYP2C9CYP2C19
SCHEMBL2907021 0.73 L3MBTL1 (0.58) ALDH1A1KDM4ECYP3A4CYP2C19CYP1A2
SCHEMBL2907654 0.73 RECQL (0.59) ALDH1A1KDM4ECYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003099812-A1 PHENYL-FURAN OR PHENYL-THIOPHENE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICINE PIERRE FABRE MEDICAMENT (FR) 2003-12-04 WO disclosed