SCHEMBL7263249

SCHEMBL7263249

CC(C)OP(=O)(COC(C)Cn1cnc2c(Cl)nc(N)nc21)OC(C)C

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.49
FAP Q12884 2/20 0.47
HSP90AB1 P08238 14/20 0.47
HSP90AA1 P07900 13/20 0.47
HDAC1 Q13547 2/20 0.44
HDAC6 Q9UBN7 2/20 0.44
HDAC4 P56524 1/20 0.44
HSP90B1 P14625 1/20 0.42
TRAP1 Q12931 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9176435 1.00 CYP3A4 (0.49) CYP3A4FAPHSP90AB1HSP90AA1HDAC1
SCHEMBL9177023 1.00 CYP3A4 (0.49) CYP3A4FAPHSP90AB1HSP90AA1HDAC1
SCHEMBL14244311 0.89 CYP3A4 (0.47) CYP3A4FAPHSP90AB1HSP90AA1HDAC1
SCHEMBL23223510 0.88 FAP (0.48) CYP3A4FAPHSP90AB1HSP90AA1HDAC1
SCHEMBL17194161 0.88 FAP (0.48) CYP3A4FAPHSP90AB1HSP90AA1HDAC1
SCHEMBL13360654 0.88 HSP90AB1 (0.44) CYP3A4HSP90AB1HSP90AA1HDAC1HDAC6
SCHEMBL8752233 0.87 HSP90AB1 (0.43) HSP90AB1HSP90AA1HDAC1HDAC6HDAC4
SCHEMBL8752184 0.87 HSP90AB1 (0.43) HSP90AB1HSP90AA1HDAC1HDAC6HDAC4
SCHEMBL6902158 0.87 CYP3A4 (0.65) CYP3A4HSP90AB1HSP90AA1HDAC1HDAC6
SCHEMBL6902140 0.87 CYP3A4 (0.65) CYP3A4HSP90AB1HSP90AA1HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6653296-B1 2-phosphonomethoxypropyl derivatives of purine and pyrimidine bases INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY OF THE ACADEMY OF SCIENCES OF THE CZECH REPUBLIC (CZ) 2003-11-25 US disclosed
US-6479673-B1 Antiretroviral enantiomeric nucleotide analogs INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY OF THE ACADEMY OF SCIENCES OF THE CZECH REPUBLIC (CZ) 2002-11-12 US disclosed
US-6057305-A Antiretroviral enantiomeric nucleotide analogs INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY OF THE ACADEMY OF SCIENCES OF THE CZECH REPUBLIC (CZ) 2000-05-02 US disclosed
EP-0654037-B1 ANTIRETROVIRAL ENANTIOMERIC NUCLEOTIDE ANALOGS ACAD OF SCIENCE CZECH REPUBLIC (CZ) 1999-05-12 EP disclosed
EP-0452935-B1 Chiral 2-(phosphonomethoxy)propyl guanines as antiviral agents ACAD OF SCIENCE CZECH REPUBLIC (CS) 1995-06-21 EP disclosed
EP-0654037-A1 ANTIRETROVIRAL ENANTIOMERIC NUCLEOTIDE ANALOGS INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY OF THE ACADEMY OF SCIENCES OF THE CZECH REPUBLIC (CZ) 1995-05-24 EP disclosed
US-5302585-A Viricides, HIV virus INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY OF THE ACADEMY OF SCIENCES OF THE CZECH REPUBLIC (CS) 1994-04-12 US disclosed
WO-1994003467-A2 ANTIRETROVIRAL ENANTIOMERIC NUCLEOTIDE ANALOGS INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY OF THE ACADEMY OF SCIENCES OF THE CZECH REPUBLIC (CZ) 1994-02-17 WO disclosed
EP-0452935-A1 Chiral 2-(phosphonomethoxy)propyl guanines as antiviral agents INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY OF THE ACADEMY OF SCIENCES OF THE CZECH REPUBLIC (CS) 1991-10-23 EP disclosed