SCHEMBL7264264

SCHEMBL7264264

COCCOC(=O)OC1=C(C)NC(C)=C(c2nnco2)C1c1ccccc1[N+](=O)[O-]

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.47
CACNA1C Q13936 5/20 0.47
KMT2A Q03164 5/20 0.47
ADORA3 P0DMS8 4/20 0.47
CYP1A2 P05177 4/20 0.47
CACNA1D Q01668 4/20 0.47
CACNA1F O60840 3/20 0.47
CACNA1S Q13698 3/20 0.47
CACNA1B Q00975 3/20 0.47
MAPT P10636 3/20 0.47
CYP3A4 P08684 3/20 0.47
CYP2C9 P11712 3/20 0.47
CYP2C19 P33261 3/20 0.47
ABCC4 O15439 2/20 0.47
ABCB11 O95342 2/20 0.47
ADORA2A P29274 2/20 0.47
ADORA1 P30542 2/20 0.47
OPRM1 P35372 2/20 0.47
SCN1A P35498 2/20 0.47
HTR2B P41595 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11000811 0.89 CACNA1C (0.54) LMNACACNA1CKMT2AADORA3CYP1A2
SCHEMBL7273125 0.85 LMNA (0.47) LMNACACNA1CKMT2AADORA3CYP1A2
SCHEMBL7272913 0.84 KMT2A (0.46) LMNACACNA1CKMT2AADORA3CYP1A2
SCHEMBL7273136 0.82 ALDH1A1 (0.41) KMT2AMAPTCYP3A4CYP2C9CYP2C19
SCHEMBL11576496 0.78 CACNA1D (0.52) LMNACACNA1CKMT2AADORA3CYP1A2
SCHEMBL11167378 0.78 CACNA1D (0.52) LMNACACNA1CKMT2AADORA3CYP1A2
SCHEMBL10866129 0.76 KMT2A (0.45) LMNACACNA1CKMT2AADORA3CYP1A2
SCHEMBL10864205 0.76 ALDH1A1 (0.34) LMNACACNA1CKMT2AADORA3CYP1A2
SCHEMBL11346454 0.75 CACNA1D (0.55) LMNACACNA1CKMT2AADORA3CYP1A2
SCHEMBL10528018 0.75 CACNA1D (0.55) LMNACACNA1CKMT2AADORA3CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0116708-A1 Substituted 1,4-dihydropyridines, method for their preparation and their use as pharmaceuticals CASSELLA Aktiengesellschaft (DE) 1984-08-29 EP disclosed