SCHEMBL7266161

SCHEMBL7266161

NC(=O)c1ccc(Sc2ccc(Cl)cc2)c(Cl)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.52
MAPT P10636 2/20 0.52
HPGD P15428 2/20 0.52
ALDH1A1 P00352 1/20 0.52
LMNA P02545 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
CHEK2 O96017 3/20 0.49
BCL2L1 Q07817 2/20 0.49
PDE7A Q13946 2/20 0.49
ICAM1 P05362 1/20 0.45
SELE P16581 1/20 0.45
PARP1 P09874 1/20 0.43
MAP4K4 O95819 2/20 0.43
POLB P06746 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8678351 0.88 ALDH1A1 (0.51) KDM4EMAPTHPGDALDH1A1LMNA
SCHEMBL4367931 0.82 SIRT2 (0.53) ALDH1A1LMNAMEN1KMT2ACHEK2
SCHEMBL6631157 0.81 CHEK2 (0.54) KDM4EMAPTHPGDALDH1A1LMNA
SCHEMBL7264564 0.80 CHEK2 (0.45) KDM4EMAPTHPGDALDH1A1LMNA
SCHEMBL5326846 0.77 HPGD (0.56) KDM4EMAPTHPGDALDH1A1LMNA
SCHEMBL2850866 0.77 BCL2L1 (0.51) KDM4EMAPTHPGDALDH1A1LMNA
SCHEMBL29503125 0.76 AR (0.53) PARP1
SCHEMBL11761622 0.74 MEN1 (0.60) KDM4EMAPTHPGDALDH1A1LMNA
SCHEMBL1149093 0.74 PDE7A (0.85) KDM4EMAPTHPGDALDH1A1LMNA
SCHEMBL2790717 0.72 HSD11B1 (0.45) CHEK2PARP1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151529-B1 5-(AMINO OR SUBSTITUTED AMINO)-1,2,3-TRIAZOLES MERCK & CO. INC. (US) 1991-09-18 EP disclosed
US-4590201-A ANTICOCCIDIAL AGENT FOR ANIMALS PARTICULARLY FOR POULTRY MERCK & CO., INC. (US) 1986-05-20 US disclosed
EP-0151529-A2 5-(Amino or substituted amino)-1,2,3-triazoles MERCK & CO. INC. (US) 1985-08-14 EP disclosed