SCHEMBL7267182

SCHEMBL7267182

COc1cc2c(cc1OC)CCC(C(N)=NO)=C2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.40
MAOA P21397 3/20 0.40
ALDH1A1 P00352 2/20 0.40
GLA P06280 2/20 0.40
GAA P10253 2/20 0.39
RECQL P46063 1/20 0.39
MAPT P10636 2/20 0.36
CYP3A4 P08684 1/20 0.36
PTGS2 P35354 1/20 0.36
ATM Q13315 2/20 0.34
TDP1 Q9NUW8 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33
HTR3A P46098 1/20 0.33
HTR3D Q70Z44 1/20 0.33
HTR3C Q8WXA8 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10715683 0.86 MAPT (0.41) KDM4EMAOAALDH1A1GLAGAA
Hydrochloric Acid SCHEMBL10715847 0.85 MAPT (0.40) KDM4EMAOAALDH1A1GLAGAA
SCHEMBL28025224 0.81 KDM4E (0.41) KDM4EMAOAALDH1A1GLAMAPT
SCHEMBL1589841 0.76 KDM4E (0.42) KDM4EMAOAALDH1A1GLAMAPT
SCHEMBL10439343 0.75 KDM4E (0.41) KDM4EMAOAALDH1A1GLAMAPT
SCHEMBL1589895 0.75 KDM4E (0.41) KDM4EMAOAALDH1A1GLAMAPT
SCHEMBL7267172 0.73 KDM4E (0.40) KDM4EMAOAALDH1A1GLAGAA
SCHEMBL10710633 0.73 HDAC1 (0.42) KDM4EMAOAALDH1A1GLAMAPT
Hydrochloric Acid SCHEMBL10800102 0.72 MAOA (0.39) KDM4EMAOAALDH1A1GLAMAPT
SCHEMBL10711338 0.72 HDAC1 (0.41) KDM4EMAOAALDH1A1GLAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0199393-B1 INDENE AND NAPHTHALENE DERIVATIVES AKZO N.V. (NL) 1988-12-07 EP claimed
US-4705782-A Indene and naphthalene derivatives AKZO N.V. (NL) 1987-11-10 US claimed
EP-0352832-B1 COMPOUNDS WITH BRONCHODILATOR ACTIVITY AKZO N.V. (NL) 1992-05-06 EP disclosed
US-5026724-A Benzothiophene derivatives AKZO N.V. (NL) 1991-06-25 US disclosed
EP-0352832-A1 Compounds with bronchodilator activity AKZO N.V. (NL) 1990-01-31 EP disclosed