SCHEMBL7267604

SCHEMBL7267604

C#CC(C)(C)OC(=O)C(O)(c1ccccc1)C1CCCCC1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.55
NFE2L2 Q16236 1/20 0.55
CHRM2 P08172 4/20 0.55
CHRM1 P11229 3/20 0.55
KCNH2 Q12809 3/20 0.55
SLC6A3 Q01959 2/20 0.55
POLB P06746 1/20 0.54
ALDH1A1 P00352 2/20 0.53
CHRM3 P20309 3/20 0.53
CYP2C19 P33261 2/20 0.53
CYP1A2 P05177 2/20 0.53
CHRM4 P08173 2/20 0.53
CHRM5 P08912 2/20 0.53
HTR2B P41595 2/20 0.53
CYP3A4 P08684 2/20 0.53
CYP2D6 P10635 2/20 0.53
CYP2C9 P11712 1/20 0.53
PKM P14618 1/20 0.53
NFKB1 P19838 1/20 0.53
THPO P40225 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7268543 0.99 KEAP1 (0.56) KEAP1NFE2L2CHRM2CHRM1KCNH2
SCHEMBL9618325 0.84 POLB (0.54) KEAP1NFE2L2CHRM2CHRM1KCNH2
SCHEMBL7915539 0.83 POLB (0.53) KEAP1NFE2L2CHRM2CHRM1KCNH2
SCHEMBL7274104 0.83 CHRM2 (0.54) KEAP1NFE2L2CHRM2CHRM1KCNH2
SCHEMBL7278370 0.81 CHRM3 (0.56) CHRM2CHRM1KCNH2SLC6A3ALDH1A1
SCHEMBL4741114 0.81 KEAP1 (0.68) KEAP1NFE2L2CHRM2CHRM1KCNH2
SCHEMBL1610849 0.81 KEAP1 (0.68) KEAP1NFE2L2CHRM2CHRM1KCNH2
SCHEMBL27483674 0.81 KEAP1 (0.68) KEAP1NFE2L2CHRM2CHRM1KCNH2
SCHEMBL6253092 0.80 CHRM2 (0.52) KEAP1NFE2L2CHRM2CHRM1KCNH2
Hydrochloric Acid SCHEMBL9878913 0.80 POLB (0.61) KEAP1NFE2L2CHRM2CHRM1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5036098-A Urogenital disorders NIPPON SHINYAKU CO., LTD. (JP) 1991-07-30 US disclosed
EP-0359311-A2 Butynylamine derivatives NIPPON SHINYAKU COMPANY, LIMITED (JP) 1990-03-21 EP disclosed