SCHEMBL7267752

SCHEMBL7267752

CC(C)(C)OC(=O)NC(Cc1ccccc1)CN1CCC[C@H]1C(=O)O

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACE P12821 1/20 0.60
KLK5 Q9Y337 1/20 0.54
ATM Q13315 1/20 0.54
CMA1 P23946 4/20 0.50
ADORA3 P0DMS8 1/20 0.49
ADORA2A P29274 1/20 0.49
ADORA2B P29275 1/20 0.49
ADORA1 P30542 1/20 0.49
APP P05067 3/20 0.48
CTSS P25774 2/20 0.47
CTSL P07711 1/20 0.47
CTSB P07858 1/20 0.47
CTSK P43235 1/20 0.47
KMT2A Q03164 1/20 0.46
F2 P00734 1/20 0.46
PRSS1 P07477 1/20 0.46
SCN9A Q15858 1/20 0.45
MAPK1 P28482 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7393230 1.00 ACE (0.60) ACEKLK5ATMCMA1ADORA3
SCHEMBL7356850 0.97 ACE (0.57) ACEKLK5ATMCMA1ADORA3
SCHEMBL10378309 0.97 ACE (0.57) ACEKLK5ATMCMA1ADORA3
SCHEMBL7269454 0.92 KLK5 (0.61) ACEKLK5ATMCMA1ADORA3
SCHEMBL8647455 0.92 KLK5 (0.61) ACEKLK5ATMCMA1ADORA3
SCHEMBL8647459 0.92 KLK5 (0.61) ACEKLK5ATMCMA1ADORA3
SCHEMBL7329010 0.89 ADORA3 (0.58) ACEKLK5ATMCMA1ADORA3
SCHEMBL8648992 0.89 ADORA3 (0.58) ACEKLK5ATMCMA1ADORA3
SCHEMBL8648996 0.89 ADORA3 (0.58) ACEKLK5ATMCMA1ADORA3
SCHEMBL5916350 0.84 ACE (0.72) ACEKLK5ATMCMA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0361341-A2 Therapeutics for aids based on inhibitors of HIV protease MILES INC. (US) 1990-04-04 EP disclosed
WO-1990000399-A1 RETROVIRAL PROTEASE BINDING PEPTIDES SMITHKLINE BECKMAN CORPORATION (US) 1990-01-25 WO disclosed
EP-0352000-A2 Retroviral protease binding peptides SMITHKLINE BEECHAM CORPORATION (US) 1990-01-24 EP disclosed