SCHEMBL8647459

SCHEMBL8647459

COC(=O)[C@@H]1CCCN1C[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 1/20 0.61
ACE P12821 2/20 0.54
ADORA3 P0DMS8 1/20 0.52
ADORA2A P29274 1/20 0.52
ADORA2B P29275 1/20 0.52
ADORA1 P30542 1/20 0.52
ATM Q13315 1/20 0.52
LTA4H P09960 2/20 0.48
CMA1 P23946 5/20 0.45
MMEL1 Q495T6 1/20 0.45
F2 P00734 1/20 0.45
PRSS1 P07477 1/20 0.45
KMT2A Q03164 1/20 0.44
CTSL P07711 1/20 0.44
SCN9A Q15858 1/20 0.44
APP P05067 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8647455 1.00 KLK5 (0.61) KLK5ACEADORA3ADORA2AADORA2B
SCHEMBL7269454 1.00 KLK5 (0.61) KLK5ACEADORA3ADORA2AADORA2B
SCHEMBL7267752 0.92 ACE (0.60) KLK5ACEADORA3ADORA2AADORA2B
SCHEMBL7393230 0.92 ACE (0.60) KLK5ACEADORA3ADORA2AADORA2B
SCHEMBL7329010 0.91 ADORA3 (0.58) KLK5ACEADORA3ADORA2AADORA2B
SCHEMBL8648992 0.91 ADORA3 (0.58) KLK5ACEADORA3ADORA2AADORA2B
SCHEMBL8648996 0.91 ADORA3 (0.58) KLK5ACEADORA3ADORA2AADORA2B
SCHEMBL7356850 0.89 ACE (0.57) KLK5ACEADORA3ADORA2AADORA2B
SCHEMBL10378309 0.89 ACE (0.57) KLK5ACEADORA3ADORA2AADORA2B
SCHEMBL16692005 0.87 MMEL1 (0.54) KLK5ACEADORA3ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0610743-B1 Aminomethylene-peptides as immunosuppressants BAYER AG (US) 1998-09-09 EP disclosed
EP-0610743-A1 Novel aminomethylene-peptides as immunosuppressants Bayer Corporation (US) 1994-08-17 EP disclosed