SCHEMBL7329010

SCHEMBL7329010

CC(C)(C)OC(=O)NC(Cc1ccccc1)CN1CCC[C@H]1C(=O)OCc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.58
ADORA2A P29274 1/20 0.58
ADORA2B P29275 1/20 0.58
ADORA1 P30542 1/20 0.58
MMEL1 Q495T6 1/20 0.55
CTSL P07711 1/20 0.53
KLK5 Q9Y337 1/20 0.52
ACE P12821 4/20 0.51
ATM Q13315 1/20 0.49
CTRB1 P17538 1/20 0.48
FKBP1A P62942 4/20 0.48
CMA1 P23946 2/20 0.47
SYK P43405 1/20 0.47
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8648996 1.00 ADORA3 (0.58) ADORA3ADORA2AADORA2BADORA1MMEL1
SCHEMBL8648992 1.00 ADORA3 (0.58) ADORA3ADORA2AADORA2BADORA1MMEL1
SCHEMBL7269454 0.91 KLK5 (0.61) ADORA3ADORA2AADORA2BADORA1MMEL1
SCHEMBL8647459 0.91 KLK5 (0.61) ADORA3ADORA2AADORA2BADORA1MMEL1
SCHEMBL8647455 0.91 KLK5 (0.61) ADORA3ADORA2AADORA2BADORA1MMEL1
SCHEMBL8547761 0.91 ADORA3 (0.53) ADORA3ADORA2AADORA2BADORA1MMEL1
SCHEMBL8547758 0.91 ADORA3 (0.53) ADORA3ADORA2AADORA2BADORA1MMEL1
SCHEMBL8547755 0.91 ADORA3 (0.53) ADORA3ADORA2AADORA2BADORA1MMEL1
SCHEMBL7267752 0.89 ACE (0.60) ADORA3ADORA2AADORA2BADORA1CTSL
SCHEMBL7393230 0.89 ACE (0.60) ADORA3ADORA2AADORA2BADORA1CTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0610743-B1 Aminomethylene-peptides as immunosuppressants BAYER AG (US) 1998-09-09 EP disclosed
EP-0610743-A1 Novel aminomethylene-peptides as immunosuppressants Bayer Corporation (US) 1994-08-17 EP disclosed
WO-1990000399-A1 RETROVIRAL PROTEASE BINDING PEPTIDES SMITHKLINE BECKMAN CORPORATION (US) 1990-01-25 WO disclosed
EP-0352000-A2 Retroviral protease binding peptides SMITHKLINE BEECHAM CORPORATION (US) 1990-01-24 EP disclosed