SCHEMBL7267783

SCHEMBL7267783

OC(CCl)CN1CCN(C(c2ccc(F)cc2)c2ccc(F)cc2)CC1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 2/20 0.64
ACHE P22303 3/20 0.59
MEN1 O00255 8/20 0.52
KMT2A Q03164 8/20 0.52
ATM Q13315 2/20 0.52
OPRM1 P35372 3/20 0.51
OPRD1 P41143 2/20 0.51
LMNA P02545 3/20 0.49
CYP2D6 P10635 2/20 0.49
HIF1A Q16665 2/20 0.49
MAPT P10636 2/20 0.49
HTR1A P08908 2/20 0.49
DRD2 P14416 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
MAPK1 P28482 1/20 0.49
THPO P40225 1/20 0.49
CACNA1G O43497 1/20 0.49
CACNA1H O95180 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL7275823 0.98 IGF1R (0.63) IGF1RACHEMEN1KMT2AATM
SCHEMBL7290611 0.94 ACHE (0.61) IGF1RACHEMEN1KMT2AATM
SCHEMBL7267603 0.86 IGF1R (0.66) IGF1RACHEMEN1KMT2AATM
SCHEMBL7266666 0.86 SLC6A9 (0.60) IGF1RMEN1KMT2AOPRM1OPRD1
SCHEMBL7276482 0.85 IGF1R (0.64) IGF1RACHEMEN1KMT2AATM
SCHEMBL7266954 0.84 KMT2A (0.71) IGF1RMEN1KMT2AATMOPRM1
SCHEMBL14355260 0.81 IGF1R (0.60) IGF1RACHEMEN1KMT2AATM
SCHEMBL7283033 0.81 CYP2D6 (0.65) IGF1RMEN1KMT2AOPRM1OPRD1
SCHEMBL7435733 0.81 IGF1R (0.60) IGF1RACHEMEN1KMT2AATM
Water SCHEMBL7290047 0.80 CYP2D6 (0.64) IGF1RMEN1KMT2AOPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE35072-E Cardiotonic agents and antiarrhythmic agents ORTHO PHARMACEUTICAL CORPORATION (US) 1995-10-24 US disclosed
US-5252569-A Cardiotonic, antiarrythmia agents ORTHO PHARMACEUTICAL CORPORATION (US) 1993-10-12 US disclosed
EP-0331511-B1 6-SUBSTITUTED PURINYL PIPERAZINE DERIVATIVES ORTHO PHARMACEUTICAL CORPORATION (US) 1993-07-28 EP disclosed
US-5215987-A Carbdiotonic agents ORTHO PHARMACEUTICAL CORPORATION (US) 1993-06-01 US disclosed
US-5164390-A Cardiac disorders ORTHO PHARMACEUTICAL CORPORATION (US) 1992-11-17 US disclosed
EP-0458459-A2 Substituted benzhydryl 2-hydroxypropyl piperazine derivatives ORTHO PHARMACEUTICAL CORPORATION (US) 1991-11-27 EP disclosed
EP-0458618-A1 6-Substituted purinyl piperazine derivatives ORTHO PHARMACEUTICAL CORPORATION (US) 1991-11-27 EP disclosed
US-5021574-A Cardiotonic agents, antiarrhythmia agents ORTHO PHARMACEUTICAL CORPORATION (US) 1991-06-04 US disclosed
US-5001127-A 4-substituted pyrazolo[3,4-d]pyrimidine derivatives ORTHO PHARMACEUTICAL CORPORATION (US) 1991-03-19 US disclosed
US-4885300-A CARDIOTONIC AND ANTIARRHYTHMIA AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1989-12-05 US disclosed
US-4876257-A 6-Substituted purinyl piperazine derivatives useful as cardiotonic and antiarrhythmic agents ORTHO PHARMACEUTICAL CORPORATION (US) 1989-10-24 US disclosed
EP-0331510-A2 4-Substituted pyrazolo[3,4-d]pyrimidine derivatives ORTHO PHARMACEUTICAL CORPORATION (US) 1989-09-06 EP disclosed