SCHEMBL7268192

SCHEMBL7268192

Cc1cn(-c2ccc3c(c2)CC(Br)C3=O)cn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.43
PSEN1 P49768 6/20 0.43
PSEN2 P49810 6/20 0.43
APH1B Q8WW43 6/20 0.43
NCSTN Q92542 6/20 0.43
APH1A Q96BI3 6/20 0.43
PSENEN Q9NZ42 6/20 0.43
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP19A1 P11511 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
MAOA P21397 2/20 0.37
MAOB P27338 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10739759 0.77 PDE3B (0.67) CYP3A4PSEN1PSEN2APH1BNCSTN
SCHEMBL9825522 0.76 PDE3B (0.60) CYP3A4PDE3BPDE3APDE4APDE4B
SCHEMBL2813793 0.76 PSEN1 (0.53) CYP3A4PSEN1PSEN2APH1BNCSTN
SCHEMBL7266092 0.74 PDE3B (0.43) CYP3A4PSEN1PSEN2APH1BNCSTN
SCHEMBL6972986 0.71 METAP1 (0.54) CYP19A1MAOAMAOB
Toluene SCHEMBL7273861 0.70 PSEN1 (0.48) CYP3A4PSEN1PSEN2APH1BNCSTN
SCHEMBL27985278 0.68 CYP1A2 (0.65) CYP3A4PSEN1PSEN2APH1BNCSTN
SCHEMBL9699737 0.67 PSEN1 (0.44) CYP3A4PSEN1PSEN2APH1BNCSTN
SCHEMBL9700832 0.67 PSEN1 (0.46) CYP3A4PSEN1PSEN2APH1BNCSTN
SCHEMBL8555030 0.66 METAP1 (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0314400-A1 Therapeutically active condensed thiadiazinones SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1989-05-03 EP claimed