SCHEMBL7269010

SCHEMBL7269010

CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)NC(Cc1ccccc1)C(=O)C(F)Cc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.55
ALOX15 P16050 1/20 0.55
CASP3 P42574 3/20 0.54
CTSD P07339 1/20 0.54
CTSB P07858 3/20 0.53
CTSK P43235 3/20 0.53
CTSL P07711 1/20 0.53
CTSS P25774 1/20 0.53
CASP7 P55210 1/20 0.52
TACR1 P25103 2/20 0.51
CAPN1 P07384 1/20 0.50
CASP1 P29466 1/20 0.49
CASP9 P55211 1/20 0.49
REN P00797 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7269151 0.92 ALDH1A1 (0.60) ALDH1A1ALOX15CASP3CTSDCTSB
SCHEMBL25287172 0.87 ECE1 (0.61) CASP3CTSDCTSBCTSKCTSL
SCHEMBL3058668 0.87 ECE1 (0.61) CASP3CTSDCTSBCTSKCTSL
SCHEMBL9416814 0.86 ALDH1A1 (0.62) ALDH1A1ALOX15CASP3CTSDCTSB
SCHEMBL23234582 0.86 ALDH1A1 (0.59) ALDH1A1ALOX15CASP3CTSDCTSB
SCHEMBL23269036 0.85 CASP3 (0.60) CASP3CTSDCTSBCTSKCTSL
SCHEMBL23268995 0.85 CASP3 (0.60) CASP3CTSDCTSBCTSKCTSL
SCHEMBL10084325 0.85 CASP3 (0.60) CASP3CTSDCTSBCTSKCTSL
SCHEMBL6269817 0.85 CTSD (0.59) ALDH1A1ALOX15CASP3CTSDCTSB
SCHEMBL8492203 0.84 CTSD (0.54) CASP3CTSDCTSBCTSKCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed