SCHEMBL7269369

SCHEMBL7269369

CCCn1c(=O)c2ncn(C34CC5CC(CC(C5)C3)C4)c2n(CCC)c1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.45
ADORA2A P29274 9/20 0.42
ADORA2B P29275 4/20 0.42
ADORA3 P0DMS8 2/20 0.42
SLC6A3 Q01959 1/20 0.42
SLC22A6 Q4U2R8 1/20 0.42
SLC22A8 Q8TCC7 1/20 0.42
SLC22A11 Q9NSA0 1/20 0.42
PDE4A P27815 7/20 0.40
PDE4B Q07343 7/20 0.40
PDE4C Q08493 7/20 0.40
PDE4D Q08499 7/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
BLM P54132 1/20 0.40
PMP22 Q01453 1/20 0.40
HSD17B10 Q99714 1/20 0.40
PI4KA P42356 1/20 0.40
PI4K2B Q8TCG2 1/20 0.40
PI4K2A Q9BTU6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10420653 0.72 PDE4A (0.49) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL3171115 0.71 ADORA2A (0.55) ADORA1ADORA2AADORA2BADORA3PDE4A
SCHEMBL9287682 0.69 ADORA2A (0.56) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL4120049 0.68 ADORA2A (0.54) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL7162120 0.67 ADORA2A (0.47) ADORA2AADORA2BADORA3PDE4APDE4B
Rolofylline SCHEMBL18029490 0.64 ADORA2A (0.71) ADORA1ADORA2AADORA2BADORA3SLC6A3
SCHEMBL7270107 0.63 ADORA1 (0.59) ADORA1ADORA2AADORA2BADORA3SLC6A3
SCHEMBL8710809 0.62 ADORA3 (0.39) ADORA1ADORA2AADORA3
SCHEMBL7269366 0.62 ADORA1 (1.00) ADORA1ADORA2AADORA2BADORA3SLC6A3
SCHEMBL7268807 0.61 ADORA2A (0.61) ADORA1ADORA2AADORA2BADORA3SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0415456-A2 Xanthine compounds KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-03-06 EP disclosed