SCHEMBL10420653

SCHEMBL10420653

CCCn1c(=O)c2ncn(N)c2n(CCC)c1=O

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 12/20 0.49
PDE4B Q07343 12/20 0.49
PDE4C Q08493 12/20 0.49
PDE4D Q08499 12/20 0.49
ADORA2A P29274 9/20 0.49
ADORA2B P29275 4/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
BLM P54132 1/20 0.49
PMP22 Q01453 1/20 0.49
HSD17B10 Q99714 1/20 0.49
PDE1A P54750 1/20 0.44
PDE1B Q01064 1/20 0.44
PDE1C Q14123 1/20 0.44
TNF P01375 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9287682 0.78 ADORA2A (0.56) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL4120049 0.77 ADORA2A (0.54) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL7162120 0.76 ADORA2A (0.47) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL3171115 0.75 ADORA2A (0.55) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL7269369 0.72 ADORA1 (0.45) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL3272841 0.71 LMNA (0.54) ADORA2AADORA2BHSD17B10
SCHEMBL8710809 0.70 ADORA3 (0.39) ADORA2A
SCHEMBL27304624 0.68 ADORA2B (0.56) ADORA2AADORA2BCYP1A2CYP3A4HSD17B10
SCHEMBL13111704 0.67 NPC1 (0.56) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL4983107 0.67 PDE4A (0.60) PDE4APDE4BPDE4CPDE4DADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4968672-A DRUG DELIVERY; DIURETICS, KIDNEY DISORDERS, HYPOTENSIVE AGENTS THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1990-11-06 US disclosed