SCHEMBL7269463

SCHEMBL7269463

CN1CCCC[C@H]1COC(=O)c1c[nH]c2ccccc12

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.60
ALDH1A1 P00352 1/20 0.60
CYP1A2 P05177 1/20 0.60
CYP2C9 P11712 1/20 0.60
TSHR P16473 1/20 0.60
THPO P40225 1/20 0.60
PMP22 Q01453 1/20 0.59
RAB9A P51151 2/20 0.57
CHRNB2 P17787 3/20 0.57
CHRNA7 P36544 3/20 0.57
CHRNA4 P43681 3/20 0.57
CHRNA5 P30532 1/20 0.57
HTR4 Q13639 2/20 0.57
NPC1 O15118 1/20 0.56
HTR6 P50406 4/20 0.53
HTR3E A5X5Y0 2/20 0.52
HTR3B O95264 2/20 0.52
HTR3A P46098 2/20 0.52
HTR3D Q70Z44 2/20 0.52
HTR3C Q8WXA8 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7269469 1.00 CYP2D6 (0.60) CYP2D6ALDH1A1CYP1A2CYP2C9TSHR
SCHEMBL7271039 1.00 CYP2D6 (0.60) CYP2D6ALDH1A1CYP1A2CYP2C9TSHR
SCHEMBL7277894 0.99 CYP2D6 (0.62) CYP2D6ALDH1A1CYP1A2CYP2C9TSHR
SCHEMBL7918881 0.97 CHRNB2 (0.61) CYP2D6ALDH1A1CYP1A2CYP2C9TSHR
SCHEMBL7918883 0.97 CHRNB2 (0.61) CYP2D6ALDH1A1CYP1A2CYP2C9TSHR
SCHEMBL7280163 0.89 CYP2D6 (0.64) CYP2D6ALDH1A1CYP1A2CYP2C9TSHR
SCHEMBL7276029 0.88 RAB9A (0.56) CYP2D6ALDH1A1CYP1A2CYP2C9TSHR
SCHEMBL7270653 0.87 CYP2D6 (0.56) CYP2D6ALDH1A1CYP1A2CYP2C9TSHR
SCHEMBL7299257 0.87 CYP2D6 (0.64) CYP2D6ALDH1A1CYP1A2CYP2C9TSHR
SCHEMBL7270646 0.86 RAB9A (0.54) CYP2D6ALDH1A1CYP1A2CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0429984-B1 Indole derivatives NISSHIN FLOUR MILLING CO (JP) 1997-07-23 EP disclosed
US-5124324-A Psychological disorders, 5-hydroxy tryptamine antagonists NISSHIN FLOUR MILLING CO., LTD. (JP) 1992-06-23 US disclosed
EP-0429984-A2 Indole derivatives NISSHIN FLOUR MILLING CO., LTD. (JP) 1991-06-05 EP disclosed