SCHEMBL7269526

SCHEMBL7269526

CC(CN1CCN(C)CC1)OC(=O)c1cn(C(=O)c2c[nH]c3ccccc23)c2ccccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
POLB P06746 1/20 0.49
ALDH1A1 P00352 3/20 0.45
PLK1 P53350 1/20 0.45
MAPT P10636 2/20 0.43
RAB9A P51151 1/20 0.43
TSHR P16473 2/20 0.43
DRD2 P14416 1/20 0.43
DRD3 P35462 1/20 0.43
HTT P42858 1/20 0.42
MAPK14 Q16539 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
THPO P40225 1/20 0.42
PMP22 Q01453 1/20 0.41
KMT2A Q03164 2/20 0.41
GAA P10253 1/20 0.41
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7297964 0.89 NPC1 (0.48) SMN1; SMN2ALDH1A1MAPTRAB9ATSHR
SCHEMBL7270889 0.87 SMN1; SMN2 (0.63) USP2SMN1; SMN2POLBALDH1A1MAPT
SCHEMBL7297419 0.85 KMT2A (0.43) SMN1; SMN2ALDH1A1MAPTRAB9ATSHR
SCHEMBL7296520 0.82 KMT2A (0.45) SMN1; SMN2ALDH1A1MAPTRAB9ATSHR
SCHEMBL7298043 0.76 NPC1 (0.61) SMN1; SMN2ALDH1A1MAPTRAB9ATSHR
SCHEMBL7297721 0.72 NPC1 (0.52) SMN1; SMN2ALDH1A1MAPTRAB9ATSHR
SCHEMBL948677 0.69 GFER (0.71) POLBALDH1A1RAB9ADRD2DRD3
SCHEMBL7298589 0.67 KMT2A (0.54) SMN1; SMN2ALDH1A1MAPTRAB9ATSHR
SCHEMBL7545507 0.67 NR4A2 (0.57) SMN1; SMN2POLBALDH1A1MAPTTSHR
SCHEMBL7288972 0.67 GABRA1 (0.47) ALDH1A1MAPTRAB9ATSHRHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0429984-B1 Indole derivatives NISSHIN FLOUR MILLING CO (JP) 1997-07-23 EP disclosed
US-5124324-A Psychological disorders, 5-hydroxy tryptamine antagonists NISSHIN FLOUR MILLING CO., LTD. (JP) 1992-06-23 US disclosed
EP-0429984-A2 Indole derivatives NISSHIN FLOUR MILLING CO., LTD. (JP) 1991-06-05 EP disclosed