SCHEMBL7297964

SCHEMBL7297964

CC1CCN(CC(C)OC(=O)c2cn(C(=O)c3c[nH]c4ccccc34)c3ccccc23)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.48
RAB9A P51151 1/20 0.48
DRD2 P14416 1/20 0.42
DRD4 P21917 1/20 0.42
DRD3 P35462 1/20 0.42
KMT2A Q03164 4/20 0.41
MEN1 O00255 3/20 0.41
TSHR P16473 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
HTR4 Q13639 2/20 0.41
HTR3E A5X5Y0 1/20 0.41
HTR3B O95264 1/20 0.41
CHRNA1 P02708 1/20 0.41
CHRNG P07510 1/20 0.41
CYP3A4 P08684 1/20 0.41
HTR1A P08908 1/20 0.41
CHRM5 P08912 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAPT P10636 1/20 0.41
CHRM1 P11229 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7297419 0.91 KMT2A (0.43) NPC1RAB9AKMT2AMEN1TSHR
SCHEMBL7269526 0.89 USP2 (0.52) RAB9ADRD2DRD3KMT2ATSHR
SCHEMBL7298043 0.88 NPC1 (0.61) NPC1RAB9ADRD2DRD4DRD3
SCHEMBL7296520 0.85 KMT2A (0.45) NPC1RAB9AKMT2AMEN1TSHR
SCHEMBL7297721 0.79 NPC1 (0.52) NPC1RAB9AKMT2AMEN1TSHR
SCHEMBL7270889 0.76 SMN1; SMN2 (0.63) RAB9ATSHRSMN1; SMN2HTR4HTR3E
SCHEMBL7298589 0.72 KMT2A (0.54) NPC1RAB9AKMT2ATSHRSMN1; SMN2
SCHEMBL7288972 0.69 GABRA1 (0.47) NPC1RAB9AKMT2ATSHRHTR4
SCHEMBL7545507 0.66 NR4A2 (0.57) KMT2AMEN1TSHRSMN1; SMN2MAPT
SCHEMBL3262552 0.64 NR4A2 (0.69) KMT2ASMN1; SMN2HTR4HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5124324-A Psychological disorders, 5-hydroxy tryptamine antagonists NISSHIN FLOUR MILLING CO., LTD. (JP) 1992-06-23 US disclosed
EP-0429984-A2 Indole derivatives NISSHIN FLOUR MILLING CO., LTD. (JP) 1991-06-05 EP disclosed