SCHEMBL7271200

SCHEMBL7271200

Cc1nc(N)nc(N)c1-c1cc(Cl)c(N)c(Cl)c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HEXA P06865 3/20 0.42
HEXB P07686 3/20 0.42
DHFR P00374 4/20 0.41
MEN1 O00255 1/20 0.38
SLC22A1 O15245 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
HTR1A P08908 1/20 0.38
ADRA2A P08913 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
HTR2A P28223 1/20 0.38
ADRA1A P35348 1/20 0.38
HTR2B P41595 1/20 0.38
SLC6A3 Q01959 1/20 0.38
KMT2A Q03164 1/20 0.38
PDE4D Q08499 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7271143 0.89 HEXA (0.42) HEXAHEXBDHFRMEN1SLC22A1
SCHEMBL6049569 0.85 DHFR (0.46) HEXAHEXBDHFRMEN1SLC22A1
Metoprine SCHEMBL29463675 0.83 NPC1 (0.54) DHFRTP53CYP1A2CYP3A4CYP2D6
Metoprine SCHEMBL3681 0.83 NPC1 (0.54) DHFRTP53CYP1A2CYP3A4CYP2D6
SCHEMBL10999078 0.81 ALDH1A1 (0.48) HEXAHEXBDHFRMEN1SLC22A1
Metoprine SCHEMBL4529657 0.81 NPC1 (0.53) DHFRTP53CYP1A2CYP3A4CYP2D6
SCHEMBL12368254 0.79 HEXA (0.64) HEXAHEXBDHFRALDH1A1RAB9A
SCHEMBL4535505 0.77 HRH4 (0.47) DHFRALDH1A1
SCHEMBL7280206 0.77 KMT2A (0.34) HEXAHEXBDHFRMEN1ALDH1A1
SCHEMBL7280211 0.77 KMT2A (0.34) HEXAHEXBDHFRMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0679645-A1 Pharmacologically active CNS pyridmidin compounds THE WELLCOME FOUNDATION LIMITED (GB) 1995-11-02 EP claimed
EP-0459819-A2 Pharmacologically active CNS compound THE WELLCOME FOUNDATION LIMITED (GB) 1991-12-04 EP claimed
EP-0679645-A1 Pharmacologically active CNS pyridmidin compounds THE WELLCOME FOUNDATION LIMITED (GB) 1995-11-02 EP disclosed
EP-0459819-A2 Pharmacologically active CNS compound THE WELLCOME FOUNDATION LIMITED (GB) 1991-12-04 EP disclosed