SCHEMBL7280206

SCHEMBL7280206

Cc1nc(N)nc(N)c1-c1cc(Cl)c(/N=C/N(C)C)c(Cl)c1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.34
HEXA P06865 1/20 0.34
HEXB P07686 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
DHFR P00374 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7280211 1.00 KMT2A (0.34) KMT2AHEXAHEXBKDM4EMEN1
SCHEMBL7272766 0.83 ALDH1A1 (0.37) KMT2AHEXAHEXBKDM4ENPC1
SCHEMBL7272773 0.83 ALDH1A1 (0.37) KMT2AHEXAHEXBKDM4ENPC1
SCHEMBL9848568 0.78 CSNK1A1 (0.41) KMT2AKDM4EALDH1A1
SCHEMBL9848576 0.78 CSNK1A1 (0.41) KMT2AKDM4EALDH1A1
SCHEMBL7271143 0.77 HEXA (0.42) KMT2AHEXAHEXBMEN1NPC1
SCHEMBL7271200 0.77 HEXA (0.42) KMT2AHEXAHEXBMEN1NPC1
SCHEMBL7280636 0.76 DHFR (0.52) KMT2AKDM4EALDH1A1DHFR
SCHEMBL6049569 0.73 DHFR (0.46) KMT2AHEXAHEXBMEN1ALDH1A1
SCHEMBL11133814 0.71 KMT2A (0.47) KMT2AKDM4EMEN1NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0679645-A1 Pharmacologically active CNS pyridmidin compounds THE WELLCOME FOUNDATION LIMITED (GB) 1995-11-02 EP disclosed
EP-0459819-A2 Pharmacologically active CNS compound THE WELLCOME FOUNDATION LIMITED (GB) 1991-12-04 EP disclosed