SCHEMBL7272095

SCHEMBL7272095

CN1[C@@H]2CC[C@H]1C[C@@H](N1C(=O)c3cccc4cccc(c34)C1=O)C2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 2/20 0.45
HPGD P15428 2/20 0.45
HSD17B10 Q99714 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
CYP1B1 Q16678 1/20 0.45
ERCC1 P07992 1/20 0.45
FEN1 P39748 1/20 0.45
ERCC4 Q92889 1/20 0.45
HTR3A P46098 1/20 0.44
ADRB2 P07550 1/20 0.43
ADRB1 P08588 1/20 0.43
ADRB3 P13945 1/20 0.43
HEXA P06865 4/20 0.43
HEXB P07686 4/20 0.43
OGA O60502 1/20 0.42
LMNA P02545 1/20 0.42
CHRNB4 P30926 1/20 0.42
CHRNA3 P32297 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7272100 1.00 ALDH1A1 (0.45) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL7281339 1.00 ALDH1A1 (0.45) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL7276878 0.94 HTR3A (0.51) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL7279088 0.94 HTR3A (0.51) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL7276880 0.94 HTR3A (0.51) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL13016514 0.87 CHRNB4 (0.44) HTR3ALMNACHRNB4CHRNA3
SCHEMBL7227680 0.85 CHRNB4 (0.50) ALDH1A1KMT2AHTR3ACHRNB4CHRNA3
SCHEMBL1573787 0.85 CHRNB4 (0.50) ALDH1A1KMT2AHTR3ACHRNB4CHRNA3
SCHEMBL3759811 0.85 CHRNB4 (0.50) ALDH1A1KMT2AHTR3ACHRNB4CHRNA3
SCHEMBL9585101 0.80 ADRB2 (0.49) ALDH1A1KDM4EHPGDHSD17B10MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5202318-A Antiserotonine, antiemetic agents SYNTEX (U.S.A.) INC. (US) 1993-04-13 US disclosed
EP-0457243-A1 Novel tricyclic compounds SYNTEX (U.S.A.) INC. (US) 1991-11-21 EP disclosed