SCHEMBL7272115

SCHEMBL7272115

COc1ccc2cc(-c3ccncn3)ccc2n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.43
CYP2D6 P10635 2/20 0.41
ADORA1 P30542 1/20 0.40
PDGFRB P09619 3/20 0.40
PDGFRA P16234 3/20 0.40
CLK1 P49759 2/20 0.40
GAK O14976 1/20 0.38
CYP19A1 P11511 1/20 0.37
CDK5 Q00535 2/20 0.36
CDK5R1 Q15078 2/20 0.36
CCNT1 O60563 1/20 0.36
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
CDK9 P50750 1/20 0.36
CCNA1 P78396 1/20 0.36
FGFR4 P22455 1/20 0.36
ROCK1 Q13464 2/20 0.36
CLK4 Q9HAZ1 2/20 0.36
GSK3B P49841 2/20 0.36
ROCK2 O75116 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7270867 0.80 PIK3CD (0.47) HPGDCYP2D6ADORA1PDGFRBPDGFRA
SCHEMBL15344999 0.77 HPGD (0.46) HPGDADORA1PDGFRBPDGFRAMAOA
SCHEMBL29941357 0.75 CYP19A1 (0.56) CYP2D6PDGFRBPDGFRACYP19A1MAPK1
SCHEMBL7270915 0.74 ADORA1 (0.42) HPGDADORA1PDGFRBPDGFRACLK1
SCHEMBL26632728 0.74 NPC1 (0.65) HPGDPDGFRBPDGFRAGSK3BCYP3A4
SCHEMBL30629466 0.74 NPC1 (0.65) HPGDPDGFRBPDGFRAGSK3BCYP3A4
SCHEMBL15341950 0.74 HPGD (0.41) HPGDADORA1PDGFRBPDGFRACLK1
SCHEMBL7264558 0.72 CYP11B2 (0.64) PDGFRBPDGFRACYP19A1CDK5CDK9
SCHEMBL12695592 0.72 BACE1 (0.57) HPGDADORA1PDGFRBPDGFRACYP19A1
SCHEMBL16573997 0.72 PDGFRB (0.46) HPGDADORA1PDGFRBPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4710507-A Quinolone inotropic agents PFIZER INC. (US) 1987-12-01 US disclosed
EP-0148623-A2 Quinolone inotropic agents Pfizer Limited (GB) 1985-07-17 EP disclosed