SCHEMBL7270915

SCHEMBL7270915

COc1ccc2cc(-c3cccnn3)ccc2n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.42
HPGD P15428 1/20 0.41
DHODH Q02127 1/20 0.39
KDM4E B2RXH2 4/20 0.38
NPC1 O15118 4/20 0.38
RAB9A P51151 4/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
ALDH1A1 P00352 2/20 0.38
POLB P06746 1/20 0.37
SLC6A2 P23975 1/20 0.36
SLC6A3 Q01959 1/20 0.36
PDE10A Q9Y233 3/20 0.36
PDE2A O00408 2/20 0.36
CYP17A1 P05093 2/20 0.35
CYP11B2 P19099 2/20 0.35
CYP19A1 P11511 1/20 0.35
CYP11B1 P15538 1/20 0.35
GSK3B P49841 1/20 0.35
DYRK1A Q13627 1/20 0.35
NFKB1 P19838 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7264558 0.75 CYP11B2 (0.64) PDE10APDE2ACYP17A1CYP11B2CYP19A1
SCHEMBL12695592 0.75 BACE1 (0.57) ADORA1HPGDKDM4ENPC1RAB9A
SCHEMBL15344999 0.74 HPGD (0.46) ADORA1HPGDNPC1RAB9APDE10A
SCHEMBL7272115 0.74 HPGD (0.43) ADORA1HPGDCYP19A1GSK3BDYRK1A
SCHEMBL7270867 0.74 PIK3CD (0.47) ADORA1HPGDCYP17A1CYP11B2CYP19A1
SCHEMBL7272193 0.74 PDGFRB (0.41) ADORA1HPGDCYP17A1CYP11B2CYP19A1
SCHEMBL7345238 0.73 PDE10A (0.52) ADORA1HPGDDHODHNPC1RAB9A
SCHEMBL16573997 0.72 PDGFRB (0.46) ADORA1HPGDNPC1RAB9APDE10A
SCHEMBL27736352 0.72 ALDH1A1 (0.50) HPGDKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL15341950 0.71 HPGD (0.41) ADORA1HPGDKDM4ENPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4710507-A Quinolone inotropic agents PFIZER INC. (US) 1987-12-01 US disclosed
EP-0148623-A2 Quinolone inotropic agents Pfizer Limited (GB) 1985-07-17 EP disclosed