SCHEMBL7273229

SCHEMBL7273229

Cn1cc(C(OC(=O)/C=C\C(=O)OC(C(=O)Cc2c[nH]cn2)c2cn(C)c3ccc(F)cc23)C(=O)Cc2c[nH]cn2)c2cc(F)ccc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
KDR P35968 4/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
CMA1 P23946 1/20 0.32
THRB P10828 1/20 0.32
MTNR1A P48039 3/20 0.32
MTNR1B P49286 3/20 0.32
EGFR P00533 2/20 0.31
HTR3A P46098 2/20 0.31
ICMT O60725 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
PER2 O15055 1/20 0.30
CRY1 Q16526 1/20 0.30
CRY2 Q49AN0 1/20 0.30
GSK3B P49841 2/20 0.30
AURKA O14965 1/20 0.30
JAK2 O60674 1/20 0.30
PAK4 O96013 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7297785 0.84 HTR3E (0.42) KDM4EALDH1A1KDRPTGDR2CMA1
SCHEMBL7272916 0.75 HTR3E (0.46) KDM4EALDH1A1MTNR1AMTNR1BHTR3A
Fumaric Acid SCHEMBL7273241 0.73 MEN1 (0.39) KDM4EALDH1A1KDRPTGDR2EGFR
Maleic Acid SCHEMBL7273221 0.73 MEN1 (0.39) KDM4EALDH1A1KDRPTGDR2EGFR
Maleic Acid SCHEMBL7273226 0.69 HTR3A (0.42) KDM4EALDH1A1KDRPTGDR2HTR3A
SCHEMBL7828711 0.63 KDM4E (0.51) KDM4EALDH1A1PTGDR2CMA1MTNR1A
SCHEMBL21661970 0.62 KDM4E (0.54) KDM4EALDH1A1KDRCMA1MTNR1A
SCHEMBL27489308 0.61 KDM4E (0.55) KDM4EALDH1A1KDRCMA1MTNR1A
SCHEMBL8360748 0.61 KDM4E (0.50) KDM4EALDH1A1KDRCMA1MTNR1A
Maleic Acid SCHEMBL7272831 0.60 HTR3E (0.42) KDM4EALDH1A1KDRPTGDR2EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4808581-A ANXIOLYTIC, ANTIEMETIC, TREATMENT OF PSYCHOLOGICAL DISORDERS GLAXO GROUP LIMITED (GB) 1989-02-28 US disclosed
EP-0276163-A2 Indole derivatives GLAXO GROUP LIMITED (GB) 1988-07-27 EP disclosed