SCHEMBL7273607

SCHEMBL7273607

COC(=O)C[C@@H]1C[C@@H](CCNc2cccc(-c3cccc(NC(=N)N)c3)c2)N(CCCc2ccccc2)C1=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.35
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
MGLL Q99685 1/20 0.35
BRAF P15056 1/20 0.34
F2 P00734 2/20 0.34
F10 P00742 1/20 0.34
PRSS1 P07477 1/20 0.34
SMYD2 Q9NRG4 1/20 0.34
LMNA P02545 2/20 0.33
MAPT P10636 2/20 0.33
CCKBR P32239 1/20 0.33
HTR2A P28223 1/20 0.33
PTGIR P43119 1/20 0.33
ITGB3 P05106 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7283072 0.92 ITGB3 (0.37) KMT2AALDH1A1MEN1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL8882502 0.92 ITGB3 (0.37) KMT2AALDH1A1MEN1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL7273665 0.90 F10 (0.39) F2F10PRSS1ITGB3ITGAV
Hydrochloric Acid SCHEMBL7283105 0.87 F2 (0.33) KMT2AALDH1A1MEN1CYP1A2CYP3A4
SCHEMBL7282011 0.86 ABCG2 (0.35) KMT2AALDH1A1MEN1CYP1A2CYP3A4
SCHEMBL7273655 0.86 SIGMAR1 (0.40) KMT2AALDH1A1MEN1CYP1A2CYP2C9
Hydrochloric Acid SCHEMBL7281102 0.79 F10 (0.51) F2F10PRSS1LMNA
SCHEMBL7275008 0.78
SCHEMBL7274585 0.78 ITGB3 (0.42) F2F10PRSS1ITGB3ITGAV
Hydrochloric Acid SCHEMBL7282118 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed