SCHEMBL7282011

SCHEMBL7282011

COC(=O)C[C@@H]1C[C@@H](CCNc2cccc(-c3ccc(C#N)cc3)c2)N(CCCc2ccccc2)C1=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 3/20 0.35
ABCB1 P08183 1/20 0.35
HPGD P15428 1/20 0.35
HTR1A P08908 1/20 0.35
DRD4 P21917 1/20 0.35
HTR2A P28223 1/20 0.35
HRH1 P35367 1/20 0.35
OPRM1 P35372 1/20 0.35
SMYD2 Q9NRG4 1/20 0.35
EP300 Q09472 4/20 0.35
BRD4 O60885 2/20 0.34
BRD2 P25440 2/20 0.34
BRD3 Q15059 2/20 0.34
MCHR1 Q99705 2/20 0.34
CHRM4 P08173 1/20 0.33
NAMPT P43490 1/20 0.33
ALDH1A1 P00352 2/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7273665 0.87 F10 (0.39)
SCHEMBL7273607 0.86 KMT2A (0.35) HTR2ASMYD2ALDH1A1LMNAMAPT
SCHEMBL7281022 0.85 CHRM4 (0.42) DRD4OPRM1MCHR1CHRM4NAMPT
SCHEMBL7273748 0.85 HTR1A (0.38) ABCG2ABCB1HPGDHTR1ADRD4
SCHEMBL7273655 0.85 SIGMAR1 (0.40) HPGDALDH1A1LMNAMAPTMEN1
SCHEMBL7278834 0.84 HTR1A (0.39) ABCG2ABCB1HPGDHTR1ACHRM4
SCHEMBL7281268 0.83 ABCB1 (0.44) ABCG2ABCB1HPGDHTR1ADRD4
SCHEMBL7282551 0.83 ABCB1 (0.44) ABCG2ABCB1HPGDHTR1ADRD4
SCHEMBL7274151 0.83 ABCB1 (0.44) ABCG2ABCB1HPGDHTR1ADRD4
SCHEMBL7274966 0.83 HRH3 (0.40) ABCG2ABCB1HPGDHTR1ADRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed