SCHEMBL7273748

SCHEMBL7273748

COC(=O)C[C@@H]1C[C@@H](CNc2ccc(-c3ccc(C#N)cc3)cc2)N(CCCc2ccccc2)C1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.38
DRD4 P21917 1/20 0.38
HTR2A P28223 1/20 0.38
HRH1 P35367 1/20 0.38
OPRM1 P35372 1/20 0.38
ALDH1A1 P00352 3/20 0.37
MAPT P10636 3/20 0.37
LMNA P02545 2/20 0.37
ABCB1 P08183 1/20 0.37
HPGD P15428 1/20 0.37
ABCG2 Q9UNQ0 1/20 0.37
MEN1 O00255 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
KMT2A Q03164 2/20 0.37
ALOX12 P18054 1/20 0.37
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7274708 0.89 CHRM4 (0.42) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL7274151 0.88 ABCB1 (0.44) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL7281268 0.88 ABCB1 (0.44) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL7282551 0.88 ABCB1 (0.44) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL7275885 0.87 EP300 (0.40) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL7275758 0.87 LSS (0.38) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL7282113 0.86 ITGB3 (0.38) ALDH1A1MAPTLMNAMEN1CYP1A2
SCHEMBL7273786 0.86 HTR1A (0.38) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL7274458 0.86 ABCB1 (0.43) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL7276410 0.85 HTR1A (0.37) HTR1ADRD4HTR2AHRH1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed