SCHEMBL7274134

SCHEMBL7274134

COc1ccc(CCNC(=O)c2ccc(C(=O)NCCc3ccccc3)cc2)cc1OC

nearest known ligand 0.85

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.85
RAB9A P51151 2/20 0.85
GAA P10253 1/20 0.77
MAPT P10636 5/20 0.72
ALDH1A1 P00352 3/20 0.72
SMN1; SMN2 Q16637 3/20 0.70
HPGD P15428 1/20 0.70
ALOX12 P18054 1/20 0.70
CA1 P00915 1/20 0.70
CA2 P00918 1/20 0.70
CA7 P43166 1/20 0.70
CA9 Q16790 1/20 0.70
CA14 Q9ULX7 1/20 0.70
MEN1 O00255 2/20 0.69
KMT2A Q03164 2/20 0.69
PLAAT3 P53816 1/20 0.68
PLAAT5 Q96KN8 1/20 0.68
PLAAT2 Q9NWW9 1/20 0.68
PLAAT4 Q9UL19 1/20 0.68
LMNA P02545 2/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29356619 0.95 ALDH1A1 (0.77) NPC1RAB9AGAAMAPTALDH1A1
SCHEMBL6270935 0.95 ALDH1A1 (0.77) NPC1RAB9AGAAMAPTALDH1A1
SCHEMBL14252956 0.92 SMN1; SMN2 (0.77) NPC1RAB9AGAAMAPTALDH1A1
SCHEMBL9312655 0.92 NPC1 (1.00) NPC1RAB9AGAAMAPTSMN1; SMN2
SCHEMBL7115429 0.90 GAA (0.70) NPC1RAB9AGAAMAPTALDH1A1
SCHEMBL28689186 0.88 GAA (0.79) NPC1RAB9AGAAMAPTALDH1A1
SCHEMBL4488518 0.88 GAA (0.79) NPC1RAB9AGAAMAPTALDH1A1
SCHEMBL30597452 0.88 GAA (0.79) NPC1RAB9AGAAMAPTALDH1A1
SCHEMBL11716101 0.88 MTNR1B (0.68) NPC1RAB9AGAAMAPTALDH1A1
SCHEMBL11717434 0.88 NPC1 (0.66) NPC1RAB9AGAAMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4885313-A 3,4-Dihydroxyphenylethylamine derivatives and their use FISONS PLC (GB) 1989-12-05 US disclosed
US-4803225-A Dihydroxy-phenethylamino compounds useful as pharmaceuticals FISONS, PLC (GB) 1989-02-07 US disclosed
US-4720586-A Substituted 3,4-dihydroxy-phenylethylamino compounds FISONS, PLC (GB) 1988-01-19 US disclosed
EP-0142283-A2 Phenylethylamines, process for their preparation and compositions containing them FISONS plc (GB) 1985-05-22 EP disclosed