SCHEMBL6270935

SCHEMBL6270935

COc1ccc(CCNC(=O)c2ccccc2)cc1OC

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.77
SMN1; SMN2 Q16637 2/20 0.77
HPGD P15428 1/20 0.77
ALOX12 P18054 1/20 0.77
GAA P10253 1/20 0.76
NPC1 O15118 1/20 0.76
RAB9A P51151 1/20 0.76
MAPK1 P28482 1/20 0.73
KMT2A Q03164 3/20 0.71
MAPT P10636 3/20 0.71
MEN1 O00255 2/20 0.71
CA1 P00915 1/20 0.70
CA2 P00918 1/20 0.70
CA7 P43166 1/20 0.70
CA9 Q16790 1/20 0.70
CA14 Q9ULX7 1/20 0.70
HTT P42858 1/20 0.68
NAMPT P43490 1/20 0.65
PKM P14618 1/20 0.65
POLB P06746 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29356619 1.00 ALDH1A1 (0.77) ALDH1A1SMN1; SMN2HPGDALOX12GAA
SCHEMBL7274134 0.95 NPC1 (0.85) ALDH1A1SMN1; SMN2HPGDALOX12GAA
SCHEMBL14252956 0.92 SMN1; SMN2 (0.77) ALDH1A1SMN1; SMN2HPGDALOX12GAA
SCHEMBL2775936 0.91 ALDH1A1 (0.69) ALDH1A1SMN1; SMN2HPGDALOX12GAA
SCHEMBL11716101 0.90 MTNR1B (0.68) ALDH1A1SMN1; SMN2HPGDALOX12GAA
SCHEMBL11717434 0.90 NPC1 (0.66) ALDH1A1SMN1; SMN2HPGDALOX12GAA
SCHEMBL7115429 0.90 GAA (0.70) ALDH1A1SMN1; SMN2HPGDALOX12GAA
SCHEMBL5726019 0.89 ALDH1A1 (0.63) ALDH1A1SMN1; SMN2HPGDALOX12GAA
SCHEMBL4488518 0.88 GAA (0.79) ALDH1A1SMN1; SMN2HPGDALOX12GAA
SCHEMBL28689186 0.88 GAA (0.79) ALDH1A1GAANPC1RAB9AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114671729-B Preparation method of aromatic ethylamine and derivative thereof 南京大学 2023-04-25 CN disclosed
CN-114671729-A Preparation method of aromatic ethylamine and derivatives thereof 南京大学 2022-06-28 CN disclosed
CN-107540596-B A kind of compound 5, the preparation method of 6- dihydroxy indole quinoline and its halogen acid salt 烟台六谛医药科技有限公司 2019-06-14 CN disclosed
CN-107540596-A A kind of preparation method of the dihydroxy indole quinoline of compound 5,6 and its halogen acid salt 烟台六谛医药科技有限公司 2018-01-05 CN disclosed
US-20130012536-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-01-10 US disclosed
US-20130012536-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-01-10 US disclosed
US-20120035179-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED 2012-02-09 US disclosed
US-20100125090-A1 Modulators of ATP-Binding Cassette Transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-05-20 US disclosed
US-20100125090-A1 Modulators of ATP-Binding Cassette Transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-05-20 US disclosed
US-7598412-B2 Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-10-06 US disclosed
US-7598412-B2 Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-10-06 US disclosed
EP-1440052-B1 BENZAMIDE DERIVATIVES AS ANTAGONISTS OF OREXIN RECEPTORS SMITHKLINE BEECHAM PLC (GB) 2005-12-14 EP disclosed
WO-1992000966-A1 N-DIMETHOXY PHENYL ALKYL-N'-IMIDAZOLYL PHENYL AMIDINE DERIVATIVES AND PROCESS THEREOF IL YANG PHARM. CO., LTD. (KR) 1992-01-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130012536-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS ABCB11, ABCB1, ABCC5 ALDH1A1 895/4885SMN1; SMN2 3617/4885HPGD 1656/4885
US-20100125090-A1 Modulators of ATP-Binding Cassette Transporters ABCB11, ABCB1, ABCC5 ALDH1A1 895/4885SMN1; SMN2 3617/4885HPGD 1656/4885
US-20120035179-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS ABCB11, ABCB1, ABCC5 ALDH1A1 895/4885SMN1; SMN2 3617/4885HPGD 1656/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.