SCHEMBL7274156

SCHEMBL7274156

C=CC[C@H]1C[C@@H](COc2ccc(-c3ccc(C#N)cc3)cc2)N(CCCc2ccccc2)C1=O

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.42
HPGD P15428 1/20 0.42
ABCG2 Q9UNQ0 1/20 0.42
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
HRH1 P35367 13/20 0.37
HTR1A P08908 1/20 0.37
DRD4 P21917 1/20 0.37
HTR2A P28223 1/20 0.37
OPRM1 P35372 1/20 0.37
HRH3 Q9Y5N1 14/20 0.36
HRH2 P25021 12/20 0.36
MAOB P27338 1/20 0.36
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7283159 1.00 ABCB1 (0.42) ABCB1HPGDABCG2MEN1KMT2A
SCHEMBL7282764 1.00 ABCB1 (0.42) ABCB1HPGDABCG2MEN1KMT2A
SCHEMBL7282205 0.97 ABCB1 (0.41) ABCB1HPGDABCG2MEN1KMT2A
SCHEMBL7285382 0.94 ABCB1 (0.43) ABCB1HPGDABCG2MEN1KMT2A
SCHEMBL7281199 0.90 SLC6A2 (0.37) ABCB1HPGDABCG2HRH1HTR1A
SCHEMBL7285068 0.90 HRH3 (0.41) MEN1KMT2AHRH1HRH3HRH2
SCHEMBL7281548 0.89 FAAH (0.36) HRH1HTR1ADRD4HTR2AOPRM1
SCHEMBL7275999 0.89 CYP19A1 (0.40) ABCB1HPGDABCG2MEN1KMT2A
SCHEMBL7283267 0.88 HPGD (0.34) ABCB1HPGDABCG2HRH1HTR1A
SCHEMBL7282767 0.88 HRH3 (0.40) ABCB1HPGDABCG2HRH1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed