SCHEMBL7283267

SCHEMBL7283267

C=CC[C@@H]1C[C@@H](COc2ccc(-c3ccc(C#N)cc3)cc2Br)N(CCCc2ccccc2)C1=O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.34
ABCB1 P08183 1/20 0.34
ABCG2 Q9UNQ0 1/20 0.34
HTR1A P08908 1/20 0.33
DRD4 P21917 1/20 0.33
HTR2A P28223 1/20 0.33
HRH1 P35367 1/20 0.33
OPRM1 P35372 1/20 0.33
DRD2 P14416 1/20 0.32
DRD3 P35462 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
MAPK1 P28482 1/20 0.31
CYP19A1 P11511 1/20 0.30
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7282767 0.91 HRH3 (0.40) HPGDABCB1ABCG2HTR1ADRD4
SCHEMBL7274497 0.88 MRGPRX4 (0.36) HPGDABCB1ABCG2HTR1ADRD4
SCHEMBL7282764 0.88 ABCB1 (0.42) HPGDABCB1ABCG2HTR1ADRD4
SCHEMBL7283159 0.88 ABCB1 (0.42) HPGDABCB1ABCG2HTR1ADRD4
SCHEMBL7274156 0.88 ABCB1 (0.42) HPGDABCB1ABCG2HTR1ADRD4
SCHEMBL7274473 0.88 HTR1A (0.37) HPGDABCB1ABCG2HTR1ADRD4
SCHEMBL7281425 0.88 CYP11B1 (0.33) HPGDABCB1ABCG2HTR1ADRD4
SCHEMBL7282205 0.86 ABCB1 (0.41) HPGDABCB1ABCG2HTR1ADRD4
SCHEMBL7282659 0.85 ABCB1 (0.36) HPGDABCB1ABCG2HTR1ADRD4
SCHEMBL7283287 0.85 CYP19A1 (0.33) HPGDABCB1ABCG2HTR1ADRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed