SCHEMBL7274342

SCHEMBL7274342

CSc1cc(-c2ccc(C#N)cc2)ccc1N

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 2/20 0.45
AAK1 Q2M2I8 1/20 0.42
KIF11 P52732 3/20 0.42
MMP3 P08254 1/20 0.41
EGLN2 Q96KS0 3/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
LIMK1 P53667 1/20 0.39
HRH3 Q9Y5N1 1/20 0.37
HRH4 Q9H3N8 2/20 0.37
HSP90AB1 P08238 1/20 0.37
ALDH1A1 P00352 2/20 0.36
PGR P06401 1/20 0.36
CYP2A6 P11509 1/20 0.36
CYP3A4 P08684 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7274539 0.85 KMT2A (0.41) ALDH1A1CYP2A6CYP3A4
SCHEMBL11528651 0.83 AAK1 (0.50) AAK1ALDH1A1CYP3A4TSHRHSD17B10
SCHEMBL3783187 0.80 AAK1 (0.48) AAK1KIF11ALDH1A1CYP3A4TSHR
SCHEMBL7285116 0.79 MMP3 (0.50) MAP4K4KIF11MMP3CA12CA1
SCHEMBL3784681 0.78 HSD17B10 (0.52) MAP4K4AAK1HSP90AB1ALDH1A1CYP3A4
SCHEMBL15156687 0.77 TDP1 (0.61) MAP4K4KIF11MMP3EGLN2CA12
SCHEMBL29655663 0.77 TDP1 (0.61) MAP4K4KIF11MMP3EGLN2CA12
SCHEMBL7272350 0.77 ACLY (0.47) KIF11MMP3ALDH1A1
SCHEMBL21388680 0.77 ALDH1A1 (0.65) MAP4K4KIF11MMP3EGLN2CA12
SCHEMBL7282985 0.74 ALDH1A1 (0.71) MAP4K4KIF11MMP3ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852192-A Cyclic urea derivatives, pharmaceutical compositions containing these compounds and processes for preparing them DR. KARL THOMAE GMBH (DE) 1998-12-22 US disclosed
US-5650424-A ANTIAGGLOMERANTS USING IMIDAZOLIDINDIONES DR. KARL THOMAE GMBH (DE) 1997-07-22 US disclosed
EP-0503548-B1 Cyclic urea derivatives, medicaments contaning them and process for their preparation THOMAE GMBH DR K (DE) 1997-06-04 EP disclosed
US-5478942-A Antiinflammatory agents, antiagglomerants KARL THOMAE GMBH (DE) 1995-12-26 US disclosed
US-5276049-A Treatment of thrombosis DR. KARL THOMAE GMBH (DE) 1994-01-04 US disclosed
EP-0503548-A1 Cyclic urea derivatives, medicaments contaning them and process for their preparation Dr. Karl Thomae GmbH (DE) 1992-09-16 EP disclosed