SCHEMBL7274497

SCHEMBL7274497

C=CC[C@@H]1C[C@@H](COc2ccc(-c3ccc(C#N)cc3)cc2C(F)(F)F)N(CCCc2ccccc2)C1=O

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 1/20 0.36
CTSS P25774 13/20 0.33
ABCB1 P08183 1/20 0.33
HPGD P15428 1/20 0.33
ABCG2 Q9UNQ0 1/20 0.33
CTSK P43235 3/20 0.32
SSTR4 P31391 1/20 0.32
HTR1A P08908 1/20 0.32
DRD4 P21917 1/20 0.32
HTR2A P28223 1/20 0.32
HRH1 P35367 1/20 0.32
OPRM1 P35372 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
RXRA P19793 1/20 0.32
RXRB P28702 1/20 0.32
RXRG P48443 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7282767 0.90 HRH3 (0.40) ABCB1HPGDABCG2HTR1ADRD4
SCHEMBL7281974 0.89 MRGPRX4 (0.40) MRGPRX4CTSSABCB1HPGDABCG2
SCHEMBL7283267 0.88 HPGD (0.34) ABCB1HPGDABCG2HTR1ADRD4
SCHEMBL7282764 0.86 ABCB1 (0.42) ABCB1HPGDABCG2HTR1ADRD4
SCHEMBL7283159 0.86 ABCB1 (0.42) ABCB1HPGDABCG2HTR1ADRD4
SCHEMBL7274156 0.86 ABCB1 (0.42) ABCB1HPGDABCG2HTR1ADRD4
SCHEMBL7273419 0.86 AR (0.39) MRGPRX4CTSSABCB1HPGDABCG2
SCHEMBL7281425 0.86 CYP11B1 (0.33) ABCB1HPGDABCG2HTR1ADRD4
SCHEMBL7282205 0.84 ABCB1 (0.41) ABCB1HPGDABCG2HTR1ADRD4
SCHEMBL7283287 0.83 CYP19A1 (0.33) ABCB1HPGDABCG2HTR1ADRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed