SCHEMBL7274909

SCHEMBL7274909

c1ccc(CC[C](Cc2cccc3ccccc23)c2ccccc2-c2ccccc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.51
CHRNA4 P43681 3/20 0.51
TDP1 Q9NUW8 1/20 0.44
MCL1 Q07820 2/20 0.43
BAD Q92934 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
CHRNB4 P30926 2/20 0.42
CHRNA3 P32297 2/20 0.42
FFAR1 O14842 1/20 0.41
AKR1B1 P15121 1/20 0.41
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
PTGER4 P35408 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP1A1 P04798 1/20 0.40
CYP1B1 Q16678 1/20 0.40
GPR52 Q9Y2T5 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7268159 0.87 CHRNB2 (0.42) CHRNB2CHRNA4TDP1MCL1BAD
SCHEMBL7267921 0.80 TDP1 (0.51) TDP1FFAR1AKR1B1KMT2AKDM4E
SCHEMBL7239901 0.77 GPR52 (0.49) TDP1L3MBTL1KMT2AKDM4EMEN1
SCHEMBL17435206 0.73 TDP1 (0.70) TDP1L3MBTL1KMT2AKDM4EMEN1
SCHEMBL5010156 0.72 CHRNB2 (0.52) CHRNB2CHRNA4TDP1MCL1BAD
SCHEMBL8804035 0.70 GPR52 (0.48) TDP1L3MBTL1KMT2AKDM4EMEN1
SCHEMBL7267678 0.70 GPR52 (0.48) TDP1KDM4ESMN1; SMN2CYP1A1CYP1B1
SCHEMBL1826164 0.68 CYP1A2 (0.52) TDP1MCL1AKR1B1KMT2AHPGD
Naphthalen-1-Yl-Methanol SCHEMBL27326059 0.68 TDP1 (0.57) CHRNB2CHRNA4TDP1L3MBTL1KMT2A
SCHEMBL28023427 0.67 GPR52 (0.56) CHRNB2CHRNA4CHRNB4CHRNA3FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0361341-A2 Therapeutics for aids based on inhibitors of HIV protease MILES INC. (US) 1990-04-04 EP claimed