SCHEMBL7276469

SCHEMBL7276469

N#Cc1ccc(-c2ccc(OC[C@@H]3C[C@H](CC(=O)O)C(=O)N3CCCc3ccccc3)cc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.45
HPGD P15428 1/20 0.45
ABCG2 Q9UNQ0 1/20 0.45
HRH1 P35367 6/20 0.41
HTR1A P08908 1/20 0.41
DRD4 P21917 1/20 0.41
HTR2A P28223 1/20 0.41
OPRM1 P35372 1/20 0.41
PPARD Q03181 2/20 0.40
PPARA Q07869 1/20 0.40
MMP2 P08253 1/20 0.40
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
TSHR P16473 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HRH3 Q9Y5N1 6/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7275504 1.00 ABCB1 (0.45) ABCB1HPGDABCG2HRH1HTR1A
SCHEMBL7273402 0.97 ABCB1 (0.44) ABCB1HPGDABCG2HRH1HTR1A
SCHEMBL7273518 0.94 ABCB1 (0.46) ABCB1HPGDABCG2HRH1HTR1A
SCHEMBL7274151 0.91 ABCB1 (0.44) ABCB1HPGDABCG2HRH1HTR1A
SCHEMBL7281268 0.91 ABCB1 (0.44) ABCB1HPGDABCG2HRH1HTR1A
SCHEMBL7282551 0.91 ABCB1 (0.44) ABCB1HPGDABCG2HRH1HTR1A
SCHEMBL7283466 0.90 PPARA (0.40) ABCB1HPGDABCG2HRH1HTR1A
Water SCHEMBL8882300 0.90 ITGB3 (0.38) PPARDPPARAALDH1A1LMNAMAPT
SCHEMBL7284836 0.90 MMP2 (0.46) HRH1PPARDPPARAMMP2HRH3
SCHEMBL7274360 0.89 ALDH1A1 (0.39) HRH1HTR1ADRD4HTR2AOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed