SCHEMBL7276624

SCHEMBL7276624

Cc1cc(N2CCN(C(=O)c3ccc4c(c3)CCC(=O)N4)CC2)cc2ccc(=O)[nH]c12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.56
NR3C1 P04150 1/20 0.56
PGR P06401 1/20 0.56
KCNH2 Q12809 1/20 0.56
PDE3B Q13370 1/20 0.56
PDE3A Q14432 1/20 0.56
CRBN Q96SW2 5/20 0.44
ALDH1A1 P00352 5/20 0.40
TSHR P16473 3/20 0.40
OGT O15294 1/20 0.40
HTT P42858 3/20 0.38
MAPK1 P28482 3/20 0.38
LMNA P02545 3/20 0.38
ALOX15 P16050 3/20 0.38
HTR1A P08908 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A3 Q01959 1/20 0.38
TP53 P04637 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
GLA P06280 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7269770 0.84 PDE3B (0.61) SLC6A4NR3C1PGRKCNH2PDE3B
SCHEMBL7274351 0.82 NR3C1 (0.64) SLC6A4NR3C1PGRKCNH2PDE3B
SCHEMBL7269908 0.80 SLC6A4 (0.78) SLC6A4NR3C1PGRKCNH2PDE3B
SCHEMBL2729628 0.78 NR3C1 (0.69) SLC6A4NR3C1PGRKCNH2PDE3B
SCHEMBL7319943 0.78 NR3C1 (0.66) SLC6A4NR3C1PGRKCNH2PDE3B
SCHEMBL11044555 0.76 KCNH2 (0.60) SLC6A4NR3C1PGRKCNH2PDE3B
SCHEMBL11046347 0.76 NR3C1 (0.62) SLC6A4NR3C1PGRKCNH2PDE3B
SCHEMBL7267767 0.76 SLC6A4 (0.72) SLC6A4NR3C1PGRKCNH2PDE3B
Iodide SCHEMBL11041065 0.75 NR3C1 (0.61) SLC6A4NR3C1PGRKCNH2PDE3B
SCHEMBL11045054 0.74 CRBN (0.62) SLC6A4NR3C1PGRKCNH2PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0370381-B1 2(1H)-quinolinone compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1995-05-10 EP disclosed
US-4988698-A Cardiovascular disorders, hypotensive agents FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-01-29 US disclosed
EP-0370381-A2 2(1H)-quinolinone compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1990-05-30 EP disclosed