SCHEMBL7274351

SCHEMBL7274351

Cc1cc(N2CCN(C(=O)c3ccc4c(c3)CCC(=O)N4)CC2)cc2c1NC(=O)CC2

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 1/20 0.64
PGR P06401 1/20 0.64
SLC6A4 P31645 1/20 0.64
KCNH2 Q12809 1/20 0.64
PDE3B Q13370 1/20 0.64
PDE3A Q14432 1/20 0.64
CRBN Q96SW2 8/20 0.48
ALDH1A1 P00352 4/20 0.44
TSHR P16473 3/20 0.44
OGT O15294 1/20 0.43
HTT P42858 3/20 0.41
MAPK1 P28482 2/20 0.41
ALOX15 P16050 2/20 0.41
TP53 P04637 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
NPSR1 Q6W5P4 1/20 0.41
GLA P06280 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
HTR1A P08908 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7269908 0.87 SLC6A4 (0.78) NR3C1PGRSLC6A4KCNH2PDE3B
SCHEMBL7267767 0.83 SLC6A4 (0.72) NR3C1PGRSLC6A4KCNH2PDE3B
SCHEMBL2729628 0.83 NR3C1 (0.69) NR3C1PGRSLC6A4KCNH2PDE3B
SCHEMBL7276624 0.82 SLC6A4 (0.56) NR3C1PGRSLC6A4KCNH2PDE3B
SCHEMBL7319943 0.82 NR3C1 (0.66) NR3C1PGRSLC6A4KCNH2PDE3B
SCHEMBL11044555 0.81 KCNH2 (0.60) NR3C1PGRSLC6A4KCNH2PDE3B
SCHEMBL11046347 0.81 NR3C1 (0.62) NR3C1PGRSLC6A4KCNH2PDE3B
Iodide SCHEMBL11041065 0.80 NR3C1 (0.61) NR3C1PGRSLC6A4KCNH2PDE3B
SCHEMBL7302842 0.79 SLC6A4 (0.67) NR3C1PGRSLC6A4KCNH2PDE3B
Vesnarinone SCHEMBL6243858 0.78 PDE3B (1.00) NR3C1PGRSLC6A4KCNH2PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0370381-B1 2(1H)-quinolinone compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1995-05-10 EP disclosed
US-4988698-A Cardiovascular disorders, hypotensive agents FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-01-29 US disclosed
EP-0370381-A2 2(1H)-quinolinone compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1990-05-30 EP disclosed