SCHEMBL7276676

SCHEMBL7276676

CCOC(=O)[C@H](Cc1cc([N+](=O)[O-])c(O)c([N+](=O)[O-])c1)NC(=O)C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
GPR35 Q9HC97 2/20 0.38
ESR1 P03372 1/20 0.38
MAPT P10636 2/20 0.36
LMNA P02545 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MAPK1 P28482 1/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
GALR2 O43603 1/20 0.36
MITF O75030 1/20 0.36
POLB P06746 1/20 0.36
HSP90AA1 P07900 1/20 0.36
HPGD P15428 1/20 0.36
XBP1 P17861 1/20 0.36
CCR6 P51684 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7638610 0.86 ALDH1A1 (0.49) ALDH1A1GPR35ESR1MAPTLMNA
SCHEMBL7283098 0.84 ALDH1A1 (0.43) ALDH1A1GPR35NPSR1
SCHEMBL7989753 0.81 ALDH1A1 (0.43) ALDH1A1MAPTLMNASMN1; SMN2KMT2A
SCHEMBL13013230 0.75 TP53 (0.52) POLBNPSR1
SCHEMBL7284208 0.75 ALDH1A1 (0.52) ALDH1A1GPR35ESR1MAPTLMNA
SCHEMBL5118162 0.75 NLRP3 (0.47) POLB
SCHEMBL5124369 0.75 TACR1 (0.41) ESR1SMN1; SMN2POLB
SCHEMBL8731461 0.75 THRB (0.51) ALDH1A1MAPTLMNASMN1; SMN2KMT2A
SCHEMBL12560474 0.74 MDM4 (0.42) ALDH1A1MAPTLMNAKMT2AL3MBTL1
SCHEMBL7274092 0.74 ALDH1A1 (0.53) ALDH1A1MAPTLMNASMN1; SMN2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5061798-A Intermediates in the formation of synthetic hormones, mimic effects of thyroid hormones; little or no effect on the heart SMITH KLINE & FRENCH LABORATORIES, LTD. (GB) 1991-10-29 US disclosed
EP-0188351-B1 CHEMICAL COMPOUNDS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-03-13 EP disclosed
US-4910305-A Containing a protected 4-hydroxyphenyl SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1990-03-20 US disclosed
US-4826876-A WITHOUT EFFECT ON HEART SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1989-05-02 US disclosed
US-4766121-A NOT AFFECTING THE HEART SMITH KLINE & FRENCH LABORATORIES LTD. (GB) 1988-08-23 US disclosed
EP-0188351-A2 Chemical compounds SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1986-07-23 EP disclosed