SCHEMBL7277406

SCHEMBL7277406

CC(C)(C)OC(=O)C[C@@H]1C[C@@H](COc2ccc(-c3ccc4cnccc4c3)cc2)NC1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.47
ITGA2B P08514 1/20 0.47
IRAK4 Q9NWZ3 13/20 0.37
FASN P49327 2/20 0.35
MKNK2 Q9HBH9 2/20 0.35
DYRK3 O43781 1/20 0.35
ROCK2 O75116 1/20 0.35
PRKD3 O94806 1/20 0.35
MAP4K4 O95819 1/20 0.35
CDK1 P06493 1/20 0.35
ROS1 P08922 1/20 0.35
PIM1 P11309 1/20 0.35
PRKACA P17612 1/20 0.35
RPS6KB1 P23443 1/20 0.35
CDK2 P24941 1/20 0.35
AKT1 P31749 1/20 0.35
CLK2 P49760 1/20 0.35
GSK3B P49841 1/20 0.35
IRAK1 P51617 1/20 0.35
RPS6KA3 P51812 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7286680 0.87 ITGB3 (0.62) ITGB3ITGA2BIRAK4GSK3B
SCHEMBL7285264 0.81 ITGB3 (0.53) ITGB3ITGA2BGPR119
SCHEMBL7285015 0.81 ITGB3 (0.49) ITGB3ITGA2BIRAK4GPR119
SCHEMBL8884076 0.81 ITGB3 (0.52) ITGB3ITGA2BGPR119
SCHEMBL7283463 0.79 ITGB3 (0.49) ITGB3ITGA2BIRAK4GPR119
Hydrochloric Acid SCHEMBL7275246 0.79 ITGB3 (0.58) ITGB3ITGA2BIRAK4GPR119
SCHEMBL7318086 0.79 ITGB3 (0.47) ITGB3ITGA2BIRAK4
SCHEMBL7323680 0.79 ITGB3 (0.47) ITGB3ITGA2BGPR119
Hydrochloric Acid SCHEMBL7275160 0.78 ITGB3 (0.58) ITGB3ITGA2BIRAK4GPR119
SCHEMBL7277677 0.78 ITGB3 (0.46) ITGB3ITGA2BIRAK4GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528369-B1 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation BOEHRINGER INGELHEIM PHARMA (DE) 1999-11-24 EP disclosed
US-5455348-A Anticoagulants Thomae, Karl (DE) 1995-10-03 US disclosed
EP-0528369-A2 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-02-24 EP disclosed